SCHEMBL24485702

SCHEMBL24485702

Cc1ncsc1COc1ccc2oc(C)c(C(=O)NC3(CO)CCOCC3)c2c1C

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.33
FFAR4 Q5NUL3 1/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPT P10636 2/20 0.32
CNR2 P34972 1/20 0.32
GAA P10253 1/20 0.32
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ADAMTS4 O75173 1/20 0.31
MMP3 P08254 1/20 0.31
MMP7 P09237 1/20 0.31
ADAM17 P78536 1/20 0.31
ADAMTS1 Q9UHI8 1/20 0.31
ADAMTS5 Q9UNA0 1/20 0.31
DGAT2 Q96PD7 3/20 0.31
ANO1 Q5XXA6 1/20 0.31
LMNA P02545 1/20 0.31
THRB P10828 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29629890 1.00 BTK (0.33) BTKFFAR4ALDH1A1MAPTCNR2
SCHEMBL24484957 0.92 BTK (0.32) BTKCNR2ADAMTS4MMP3MMP7
SCHEMBL29630025 0.92 BTK (0.32) BTKCNR2ADAMTS4MMP3MMP7
SCHEMBL24484331 0.90 SCN9A (0.31) BTK
SCHEMBL24484858 0.86 GABRA1 (0.32) LMNAGABRA1
SCHEMBL29629758 0.86 GABRA1 (0.32) LMNAGABRA1
SCHEMBL24484370 0.85 BTK (0.33) BTKALDH1A1MAPTCNR2GAA
SCHEMBL24484786 0.85 GAA (0.42) MAPTGAASMN1; SMN2ADAMTS4MMP3
SCHEMBL24484862 0.84
SCHEMBL29629942 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022112352-A1 HETEROCYCLE DERIVATIVES FOR TREATING TRPM3 MEDIATED DISORDERS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2022-06-02 WO disclosed