Oxethazaine

Oxethazaine

SCHEMBL24489

CN(C(=O)CN(CCO)CC(=O)N(C)C(C)(C)Cc1ccccc1)C(C)(C)Cc1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 1.00
MEN1 O00255 3/20 1.00
HIF1A Q16665 2/20 1.00
CYP3A4 P08684 2/20 1.00
CYP2C19 P33261 2/20 1.00
LMNA P02545 1/20 1.00
CYP2D6 P10635 1/20 1.00
ALOX15 P16050 1/20 1.00
TSHR P16473 1/20 1.00
SCN1A P35498 1/20 1.00
SCN2A Q99250 1/20 1.00
SCN3A Q9NY46 1/20 1.00
NPY5R Q15761 1/20 0.46
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
RIPK1 Q13546 1/20 0.36
ALDH1A1 P00352 3/20 0.36
RECQL P46063 1/20 0.36
MMP8 P22894 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxethazaine SCHEMBL4280369 1.00 KMT2A (1.00) KMT2AMEN1HIF1ACYP3A4CYP2C19
Oxethazaine SCHEMBL945710 0.99 MEN1 (0.97) KMT2AMEN1HIF1ACYP3A4CYP2C19
SCHEMBL13934977 0.95 TSHR (0.90) KMT2AMEN1HIF1ACYP3A4CYP2C19
Oxethazaine SCHEMBL18741042 0.94 CYP3A4 (0.88) KMT2AMEN1HIF1ACYP3A4CYP2C19
Oxethazaine SCHEMBL18741053 0.88 LMNA (0.78) KMT2AMEN1HIF1ACYP3A4CYP2C19
SCHEMBL9234745 0.77 KMT2A (0.62) KMT2AMEN1HIF1ACYP3A4CYP2C19
SCHEMBL7435206 0.75 CYP3A4 (0.59) KMT2AMEN1HIF1ACYP3A4CYP2C19
SCHEMBL7435200 0.73 CYP3A4 (0.57) KMT2AMEN1HIF1ACYP3A4CYP2C19
SCHEMBL23364816 0.70 MEN1 (0.53) KMT2AMEN1HIF1ACYP3A4CYP2C19
SCHEMBL18379359 0.69 LMNA (0.52) KMT2AMEN1HIF1ACYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3456 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260115156-A1 INJECTABLE COMPOSITION INCLUDING HYDROGEL CONTAINING ANESTHETIC AGENT UNIV KOREA RES & BUS FOUND (KR) 2026-04-30 US claimed
EP-4722714-A1 SIMULTANEOUS ANALYSIS OF FOOD-BORNE DOPING SUBSTANCES USING LIQUID CHROMATOGRAPHY-MASS SPECTROMETRY (VFD: VACCINE FOR FOODBORNE DOPING) Korea Institute of Science and Technology (KR) 2026-04-08 EP claimed
EP-4436552-B1 GASTRO-RETENTIVE ORAL DOSAGE UNIT CONTAINING A LOCAL ANAESTHETIC OREXA B V (NL) 2026-02-04 EP claimed
WO-2025235864-A1 COATED NEEDLE ADMINISTRATION SYSTEMS EVOLUS, INC. (US) 2025-11-13 WO claimed
US-20250319025-A9 COMPOSITIONS COMPRISING MODIFIED PHOSPHOLIPIDS AND USES THEREOF THE CHILDREN'S MEDICAL CENTER CORPORATION (US) 2025-10-16 US claimed
EP-4578441-A1 TREATMENT OF LOCALIZED PAIN PlantTec Medical GmbH (DE) 2025-07-02 EP claimed
US-20250205278-A1 METHODS AND COMPOSITIONS FOR WOUND HEALING ABBOTT NICHOLAS L (US) 2025-06-26 US claimed
WO-2025128639-A1 HYDROGELS COMPRISING PROTEIN-STABILIZED NANOPARTICLES FOR EXTENDED RELEASE THE CHILDREN'S MEDICAL CENTER CORPORATION (US) 2025-06-19 WO claimed
US-12329856-B2 Crosslinked hyaluronic acid composition with local anesthetics BIOPOLIMERI S.R.L. (IT) 2025-06-17 US claimed
US-20250186364-A1 COMBINATION OF ANTISPASMODIC AND ANESTHETIC AGENTS FOR TOPICAL PRODUCTS AND THEIR METHOD OF USE PRIMA INNOVATIONS, LLC 2025-06-12 US claimed
EP-0814773-A1 PECTIN LIQUID PHARMACEUTICAL COMPOSITIONS The Boots Company PLC (GB) 1998-01-07 EP claimed
WO-1997044021-A1 PHARMACEUTICAL PRODUCTS CONTAINING A COMPLEX OF AN AMIDE-TYPE LOCAL ANESTHETIC AND A POLYACRYLATE RHODES JOHN (GB) 1997-11-27 WO claimed
WO-1996029055-A1 PECTIN LIQUID PHARMACEUTICAL COMPOSITIONS THE BOOTS COMPANY PLC (GB) 1996-09-26 WO claimed
WO-1996029054-A1 PECTIN PHARMACEUTICAL COMPOSITIONS THE BOOTS COMPANY PLC (GB) 1996-09-26 WO claimed
US-5254591-A Oxethazaine in alginate carrier which floats on gastric fluids THE UNIVERSITY OF MELBOURNE (AU) 1993-10-19 US claimed
US-5036057-A Anesthetics THE UNIVERSITY OF MELBOURNE (AU) 1991-07-30 US claimed
EP-0250572-A1 GASTRO-OESOPHAGEAL REFLUX COMPOSITION THE UNIVERSITY OF MELBOURNE (AU) 1988-01-07 EP claimed
WO-1987004077-A1 GASTRO-OESOPHAGEAL REFLUX COMPOSITION THE UNIVERSITY OF MELBOURNE (AU) 1987-07-16 WO claimed
US-4137327-A Process for weight reduction MARSHALL EDWARD M 1979-01-30 US claimed
US-4127622-A ETHYLCELLULOSE SHELL EISAI CO., LTD. (JP) 1978-11-28 US claimed