SCHEMBL2451004

SCHEMBL2451004

CN1CCN(c2nc(-c3ccccc3C(F)(F)F)cc(NC(=O)c3cc[nH]n3)c2[N+](=O)[O-])CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 6/20 0.41
CYP1A2 P05177 4/20 0.40
CYP2D6 P10635 4/20 0.40
CYP3A4 P08684 3/20 0.40
MAPK1 P28482 2/20 0.40
SCN9A Q15858 1/20 0.39
CYP2C19 P33261 3/20 0.39
MEN1 O00255 2/20 0.38
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 2/20 0.38
CNR2 P34972 1/20 0.38
USP2 O75604 1/20 0.38
TSHR P16473 1/20 0.38
HIF1A Q16665 1/20 0.38
PTGES O14684 1/20 0.37
MAPT P10636 2/20 0.37
GAA P10253 1/20 0.37
GPR55 Q9Y2T6 1/20 0.37
SIRT6 Q8N6T7 2/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2445371 0.81 NPSR1 (0.45) WDR5CYP1A2CYP2D6CYP3A4MAPK1
SCHEMBL2444689 0.77 CYP1A2 (0.49) CYP1A2CYP2D6CYP3A4MAPK1CYP2C19
SCHEMBL2452601 0.71 CYP1A2 (0.37) CYP1A2CYP2D6CYP3A4MAPK1CYP2C19
SCHEMBL18939276 0.70 HTT (0.56) MEN1ALDH1A1KMT2ACNR2TSHR
SCHEMBL2446534 0.67 NPSR1 (0.47) SCN9AMEN1KMT2AMAPTGAA
SCHEMBL2449017 0.66 CNR2 (0.48) CYP1A2CYP2D6CYP3A4MAPK1CYP2C19
SCHEMBL2442786 0.66 MAPT (0.38) CYP1A2CYP3A4SCN9ACYP2C19MEN1
SCHEMBL14471486 0.65 CYP1A2 (0.48) CYP1A2CYP2D6CYP3A4MAPK1CYP2C19
SCHEMBL4201444 0.63 ALOX15 (0.51) CYP1A2CYP2D6CYP2C19MAPT
SCHEMBL2450125 0.61 NPSR1 (0.46) MEN1KMT2AMAPTRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011109587-A1 SUBSTITUTED AZA-BICYCLIC IMIDAZOLE DERIVATIVES USEFUL AS TRPM8 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-09-09 WO disclosed