SCHEMBL2452601

SCHEMBL2452601

Cc1nc(-c2ccccc2C(F)(F)F)nc(NC(=O)c2cc[nH]n2)c1[N+](=O)[O-]

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 6/20 0.37
CYP3A4 P08684 5/20 0.37
CYP2D6 P10635 3/20 0.37
TSHR P16473 3/20 0.37
CRHR1 P34998 1/20 0.37
CYP2C19 P33261 5/20 0.37
RECQL P46063 1/20 0.37
USP2 O75604 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.35
USP1 O94782 5/20 0.35
WDR48 Q8TAF3 5/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 4/20 0.35
MEN1 O00255 2/20 0.35
HTT P42858 2/20 0.35
KMT2A Q03164 2/20 0.35
MAPK1 P28482 1/20 0.35
NTRK1 P04629 1/20 0.34
ADORA3 P0DMS8 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2451920 0.77 NPSR1 (0.46) GAAMAPTMEN1KMT2ANTRK1
SCHEMBL2446363 0.76 AAK1 (0.38) CYP1A2CYP3A4CYP2D6CYP2C19RECQL
SCHEMBL14472097 0.73 PARP1 (0.38) CYP1A2CYP3A4CYP2D6TSHRCRHR1
SCHEMBL2442498 0.72 DPP4 (0.40) CYP1A2CYP3A4CYP2D6TSHRCRHR1
SCHEMBL2451004 0.71 WDR5 (0.41) CYP1A2CYP3A4CYP2D6TSHRCYP2C19
SCHEMBL18939276 0.69 HTT (0.56) TSHRSMN1; SMN2GAAMAPTMEN1
SCHEMBL904650 0.67 LDHA (0.46) CYP1A2CYP3A4CYP2D6TSHRCRHR1
SCHEMBL14941196 0.65 LDHA (0.41) CRHR1SMN1; SMN2MAPTMEN1HTT
SCHEMBL805590 0.63 HSD11B1 (0.51) CYP1A2CYP3A4CYP2D6TSHRCYP2C19
SCHEMBL802782 0.62 GSK3A (0.46) CYP1A2CYP3A4CYP2D6TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011109587-A1 SUBSTITUTED AZA-BICYCLIC IMIDAZOLE DERIVATIVES USEFUL AS TRPM8 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-09-09 WO disclosed