SCHEMBL2451380

SCHEMBL2451380

O=C1CCC2(CCCCC2)C(=O)O1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.38
CDC7 O00311 1/20 0.31
DBF4 Q9UBU7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4998283 0.98 TSHR (0.39) TSHR
SCHEMBL595648 0.79
SCHEMBL347199 0.76
SCHEMBL8621409 0.69 TSHR (0.43) TSHR
SCHEMBL22109759 0.69 TSHR (0.43) TSHR
SCHEMBL22470021 0.67 ALDH1A1 (0.33) CDC7DBF4
SCHEMBL15155134 0.67 CA1 (0.61) TSHR
SCHEMBL8047024 0.67 CA1 (0.50) TSHR
SCHEMBL11366827 0.67 CA1 (0.50) TSHR
SCHEMBL6283784 0.67 TSHR (0.41) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732899-B1 PROCESS FOR PREPARING CYCLOHEXANEDIACETIC ACID MONOAMIDE SERICHIM S R L (IT) 2011-09-21 EP disclosed
US-7381823-B2 Process for preparing cyclohexanediacetic acid monoamide SERICHIM S.R.L. (IT) 2008-06-03 US disclosed
US-20070208175-A1 PROCESS FOR PREPARING CYCLOHEXANEDIACETIC ACID MONOAMIDE SERICHIM S.R.L. (IT) 2007-09-06 US disclosed
EP-1753733-A1 SMALL MOLECULES FOR TREATMENT OF HYPERCHOLESTEROLEMIA AND RELATED DISEASES Avanir Pharmaceuticals (US) 2007-02-21 EP disclosed
EP-1732899-A2 PROCESS FOR PREPARING CYCLOHEXANEDIACETIC ACID MONOAMIDE SERICHUM S.R.L. (IT) 2006-12-20 EP disclosed
WO-2005123700-A1 SMALL MOLECULES FOR TREATMENT OF HYPERCHOLESTEROLEMIA AND RELATED DISEASES AVANIR PHARMACEUTICALS (US) 2005-12-29 WO disclosed
WO-2005090310-A2 PROCESS FOR PREPARING CYCLOHEXANEDIACETIC ACID MONOAMIDE SERICHIM S.R.L. (IT) 2005-09-29 WO disclosed
US-5369110-A Hypotensive agents, cardiac insufficiency treatment CIBA-GEIGY CORPORATION (US) 1994-11-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070208175-A1 PROCESS FOR PREPARING CYCLOHEXANEDIACETIC ACID MONOAMIDE GNPAT, GMDS, PIGS TSHR 4706/4885CDC7 859/4885DBF4 1355/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.