SCHEMBL24520101

SCHEMBL24520101

O=C1CN(C(=O)c2ccc(-c3ccc4ncc(C#Cc5ccnc6[nH]ccc56)n4n3)cc2)CCN1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 15/20 0.44
MKNK2 Q9HBH9 15/20 0.44
CYP3A4 P08684 1/20 0.44
EIF4E P06730 7/20 0.41
CHEK1 O14757 1/20 0.39
PIK3CA P42336 1/20 0.39
ATR Q13535 1/20 0.39
JAK2 O60674 1/20 0.39
PARP1 P09874 1/20 0.35
PARP2 Q9UGN5 1/20 0.35
KCNH2 Q12809 2/20 0.35
CCNT1 O60563 1/20 0.35
CDK9 P50750 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16626057 0.91 MKNK1 (0.55) MKNK1MKNK2CYP3A4EIF4ECHEK1
SCHEMBL16621059 0.88 CECR2 (0.47) MKNK1MKNK2CYP3A4EIF4ECHEK1
SCHEMBL16620611 0.87 MKNK1 (0.53) MKNK1MKNK2CYP3A4EIF4ECHEK1
SCHEMBL16620577 0.83 MKNK1 (0.42) MKNK1MKNK2CYP3A4EIF4ECHEK1
SCHEMBL29756310 0.80 CHEK1 (0.38) MKNK1MKNK2CYP3A4EIF4ECHEK1
SCHEMBL24520016 0.77 CHEK1 (0.42) CHEK1PIK3CAATR
SCHEMBL17969583 0.76 MET (0.41) CHEK1PIK3CAATRJAK2CDK9
SCHEMBL16625991 0.76 MKNK1 (0.52) MKNK1MKNK2CYP3A4EIF4EPIK3CA
SCHEMBL24520103 0.76 CHEK1 (0.41) CHEK1PIK3CAATRJAK2CDK9
SCHEMBL16625805 0.76 MKNK1 (0.53) MKNK1MKNK2CYP3A4EIF4EKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052501-B1 BICYCLIC ALKYNE DERIVATIVES AND USES THEREOF AGENCY SCIENCE TECH & RES (SG) 2022-06-22 EP disclosed