SCHEMBL2452120

SCHEMBL2452120

C[C@H]1C[C@@H](c2nc(-c3ccc(C#Cc4ccc5[nH]c([C@@H]6C[C@H](C)CN6C(=O)OC(C)(C)C)nc5c4)cc3)c[nH]2)N(C(=O)O)C1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.34
KCNH2 Q12809 1/20 0.34
UCHL1 P09936 1/20 0.31
HCRTR1 O43613 3/20 0.31
HCRTR2 O43614 3/20 0.31
GABRA1 P14867 2/20 0.30
GABRG2 P18507 2/20 0.30
GABRB3 P28472 2/20 0.30
GABRA3 P34903 2/20 0.30
GABRA2 P47869 2/20 0.30
PRCP P42785 1/20 0.30
PARP1 P09874 1/20 0.30
BACE1 P56817 1/20 0.30
AURKA O14965 1/20 0.30
PDPK1 O15530 1/20 0.30
AURKB Q96GD4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14849158 0.97 CYP2C9 (0.35) CYP2C9KCNH2UCHL1HCRTR1HCRTR2
SCHEMBL2448912 0.92 CYP2C9 (0.35) CYP2C9KCNH2UCHL1HCRTR1HCRTR2
SCHEMBL2450986 0.89 CYP2C9 (0.32) CYP2C9KCNH2PRCPBACE1
SCHEMBL12332958 0.88 CYP2C9 (0.37) CYP2C9KCNH2UCHL1HCRTR1HCRTR2
SCHEMBL14841446 0.88 CYP2C9 (0.37) CYP2C9KCNH2UCHL1HCRTR1HCRTR2
SCHEMBL14851380 0.88 CYP2C9 (0.37) CYP2C9KCNH2UCHL1HCRTR1HCRTR2
SCHEMBL14841447 0.88 CYP2C9 (0.37) CYP2C9KCNH2UCHL1HCRTR1HCRTR2
SCHEMBL2450982 0.86 CYP2C9 (0.30) CYP2C9KCNH2
SCHEMBL12332889 0.85 CYP2C9 (0.33) CYP2C9KCNH2PRCPPARP1BACE1
SCHEMBL10121574 0.85 PRCP (0.36) HCRTR1HCRTR2PRCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8779156-B2 Analogues for the treatment or prevention of flavivirus infections VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-07-15 US disclosed
US-20130090351-A1 ANALOGUES FOR THE TREATMENT OR PREVENTION OF FLAVIVIRUS INFECTIONS VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-04-11 US disclosed
EP-2550267-A1 ANALOGUES FOR THE TREATMENT OR PREVENTION OF FLAVIVIRUS INFECTIONS Vertex Pharmaceuticals Incorporated (US) 2013-01-30 EP disclosed
WO-2011119853-A1 ANALOGUES FOR THE TREATMENT OR PREVENTION OF FLAVIVIRUS INFECTIONS VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-09-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130090351-A1 ANALOGUES FOR THE TREATMENT OR PREVENTION OF FLAVIVIRUS INFECTIONS BLVRB, RRP1B, C1QBP CYP2C9 2576/4885KCNH2 2848/4885UCHL1 4794/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.