SCHEMBL24521443

SCHEMBL24521443

O=C(CI)N1CCC(N2CCn3nccc3C2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
KDM4E B2RXH2 5/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
ACHE P22303 3/20 0.37
ALDH1A1 P00352 4/20 0.36
MAPT P10636 2/20 0.36
HIF1A Q16665 1/20 0.36
L3MBTL3 Q96JM7 7/20 0.35
L3MBTL1 Q9Y468 5/20 0.35
TDP1 Q9NUW8 2/20 0.35
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MBTD1 Q05BQ5 4/20 0.35
TP53BP1 Q12888 1/20 0.35
L3MBTL4 Q8NA19 1/20 0.35
CBX7 O95931 2/20 0.34
CDYL2 Q8N8U2 2/20 0.34
CDYL Q9Y232 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18909452 0.87 ACACB (0.42) JAK2JAK1KDM4ECYP2C9CYP2C19
SCHEMBL22030477 0.84 FAAH (0.43) JAK2JAK1KDM4ECYP2C9CYP2C19
SCHEMBL15998855 0.68 BLM (0.43) MAPT
SCHEMBL25430636 0.67 RIPK1 (0.46)
SCHEMBL17926162 0.65 MYT1 (0.42) ALDH1A1
SCHEMBL18724894 0.65 MYT1 (0.42) CYP2C9ALDH1A1TDP1
SCHEMBL18909108 0.64 ACACB (0.42) KDM4ECYP2C9CYP2C19ACHEL3MBTL3
SCHEMBL20743163 0.64 KDR (0.38) JAK2KDM4ECYP2C9CYP2C19ACHE
SCHEMBL18909109 0.63 KDM6B (0.40) ACHE
SCHEMBL30519741 0.63 MAPK1 (0.41) ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3596072-B1 PYRAZOLOCHLOROPHENYL COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF HOFFMANN LA ROCHE (CH) 2022-06-22 EP disclosed