SCHEMBL24522243

SCHEMBL24522243

FC1(F)CCN(Cc2ccc(I)cc2)C1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.46
HRH3 Q9Y5N1 2/20 0.43
HIF1A Q16665 1/20 0.40
EPAS1 Q99814 1/20 0.40
GRM2 Q14416 1/20 0.40
HTR2A P28223 1/20 0.40
JAK2 O60674 1/20 0.39
TLR7 Q9NYK1 2/20 0.39
CYP3A4 P08684 1/20 0.38
HSD17B10 Q99714 1/20 0.38
FAAH O00519 1/20 0.38
CCR5 P51681 1/20 0.37
KDM1A O60341 1/20 0.37
MAOB P27338 1/20 0.37
RCOR1 Q9UKL0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22878453 0.85 HIF1A (0.41) SIGMAR1HRH3HIF1AEPAS1HTR2A
SCHEMBL28885908 0.83 GRM2 (0.45) SIGMAR1HRH3GRM2JAK2TLR7
SCHEMBL12176281 0.83 ALDH1A1 (0.51) SIGMAR1HRH3
SCHEMBL25181316 0.83 PRMT6 (0.45) HRH3GRM2JAK2TLR7CYP3A4
SCHEMBL3400443 0.83 ALDH1A1 (0.53) HRH3GRM2JAK2TLR7
SCHEMBL3992623 0.82 CYP3A4 (0.56) SIGMAR1HIF1ACYP3A4HSD17B10
Hydrochloric Acid SCHEMBL25412712 0.81 CYP3A4 (0.54) SIGMAR1HIF1ACYP3A4HSD17B10
SCHEMBL12074618 0.80 ALDH1A1 (0.48) HRH3GRM2JAK2TLR7FAAH
SCHEMBL25184780 0.79 USP2 (0.58) HIF1ACYP3A4HSD17B10KDM1A
SCHEMBL2558372 0.79 HRH3 (0.40) HRH3GRM2JAK2TLR7KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4015504-A1 C5AR ANTAGONISTS ChemoCentryx, Inc. (US) 2022-06-22 EP disclosed