SCHEMBL24528554

SCHEMBL24528554

Cc1ccc(O)cc1C#C[Si](C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.38
ESR2 Q92731 7/20 0.36
ESR1 P03372 6/20 0.36
CYP3A4 P08684 2/20 0.35
TSHR P16473 2/20 0.35
RECQL P46063 1/20 0.35
TTR P02766 1/20 0.34
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C9 P11712 2/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
MEN1 O00255 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B3 P37058 2/20 0.33
CA12 O43570 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15462385 0.82 NR1H3 (0.43) ESR2ESR1CYP3A4TSHRRECQL
SCHEMBL2806709 0.77 ALDH1A1 (0.45) CYP3A4TSHRRECQLTTRKDM4E
SCHEMBL14790415 0.77 KDM4E (0.33) CYP3A4TSHRKDM4EALDH1A1CYP1A2
SCHEMBL30444035 0.76 HSD17B10 (0.43) ESR2ESR1CYP3A4TSHRTTR
SCHEMBL20536435 0.76 HSD17B10 (0.43) ESR2ESR1CYP3A4TSHRTTR
SCHEMBL11296185 0.75 CSF1R (0.46) TSHRKDM4EALDH1A1CYP2C9HPGD
SCHEMBL2890025 0.74 KDM4E (0.35) CYP3A4TSHRKDM4EALDH1A1CYP1A2
SCHEMBL16620701 0.74 FFAR1 (0.47) TSHRALDH1A1GRM5
SCHEMBL4505600 0.74 TSHR (0.34) TSHRRECQLKDM4EALDH1A1HPGD
SCHEMBL16709385 0.73 ALDH1A1 (0.38) TSHRKDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129913-A1 ALKYNE DERIVATIVES AS INHIBITORS OF C-ABL BENEVOLENTAI BIO LIMITED (GB) 2022-06-23 WO disclosed