SCHEMBL24528630

SCHEMBL24528630

C=NN(c1ccccc1)c1nc(-c2ccc(/C=N/CCCN(C)C)cc2)nc(-c2ccc(/C=N\CCCN(C)C)cc2)c1C

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
LMNA P02545 1/20 0.33
RAD52 P43351 1/20 0.32
HTR7 P34969 1/20 0.32
KDM4E B2RXH2 1/20 0.31
THRB P10828 1/20 0.30
NPY1R P25929 1/20 0.30
NPY2R P49146 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
POLB P06746 1/20 0.30
HPGD P15428 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24528614 0.97 RAD52 (0.32) ALDH1A1LMNARAD52HTR7
SCHEMBL24528668 0.96 RAD52 (0.32) ALDH1A1LMNARAD52HTR7
SCHEMBL24528606 0.83 ALDH1A1 (0.34) ALDH1A1LMNAKDM4EMAPK1
SCHEMBL24528691 0.80 PDE5A (0.35) RAD52
SCHEMBL24528712 0.80 ALDH1A1 (0.34) ALDH1A1LMNAKDM4EHPGDNPSR1
SCHEMBL24528628 0.73 ADORA2A (0.34) ALDH1A1LMNARAD52POLBMAPK1
SCHEMBL24528664 0.71 ADORA2A (0.34) ALDH1A1LMNAKDM4E
SCHEMBL24528512 0.70 KDM4E (0.37) ALDH1A1LMNARAD52KDM4ETHRB
SCHEMBL29680746 0.70 KDM4E (0.37) ALDH1A1LMNARAD52KDM4ETHRB
SCHEMBL24528631 0.70 RAD52 (0.36) ALDH1A1LMNARAD52KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed