SCHEMBL24528628

SCHEMBL24528628

CN(C)CCC/N=C\c1ccc(-c2nc(-c3ccc(/C=N/CCCN(C)C)cc3)nc3ccsc23)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.34
ADORA1 P30542 7/20 0.34
ALDH1A1 P00352 2/20 0.33
LMNA P02545 1/20 0.33
PIK3CA P42336 2/20 0.33
MTOR P42345 1/20 0.33
PDGFRB P09619 1/20 0.33
KIT P10721 1/20 0.33
FLT3 P36888 1/20 0.33
PDE4A P27815 2/20 0.32
PDE4B Q07343 2/20 0.32
PDE4C Q08493 2/20 0.32
PDE4D Q08499 2/20 0.32
RAD52 P43351 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA2B P29275 1/20 0.32
POLB P06746 1/20 0.31
MAPK1 P28482 1/20 0.31
NMT1 P30419 2/20 0.31
TLR9 Q9NR96 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24528590 0.88 ADORA2A (0.40) ADORA2AADORA1ALDH1A1LMNAADORA3
SCHEMBL24528591 0.85 SCN9A (0.41) ADORA2AADORA1RAD52
SCHEMBL24528664 0.83 ADORA2A (0.34) ADORA2AALDH1A1LMNA
SCHEMBL29681009 0.82 KDM4E (0.40) ALDH1A1PIK3CAMTORPDGFRBKIT
SCHEMBL24528587 0.82 KDM4E (0.40) ALDH1A1PIK3CAMTORPDGFRBKIT
SCHEMBL24528588 0.78 ALDH1A1 (0.36) ALDH1A1PIK3CAMTORPDGFRBKIT
SCHEMBL24528709 0.73 KDM4E (0.33) ALDH1A1LMNA
SCHEMBL29680934 0.73 KDM4E (0.33) ALDH1A1LMNA
SCHEMBL24528643 0.73 NUDT1 (0.38) ALDH1A1LMNA
SCHEMBL24528630 0.73 ALDH1A1 (0.33) ALDH1A1LMNARAD52POLBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed