SCHEMBL24528632

SCHEMBL24528632

O=Cc1ccc(-c2cc(-c3ccc(C=O)cc3)c3cc[nH]c3n2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.39
CDK8 P49336 2/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C8 P10632 1/20 0.38
TGFBR1 P36897 1/20 0.38
JAK1 P23458 11/20 0.37
IKBKB O14920 3/20 0.37
CHUK O15111 3/20 0.37
DAPK3 O43293 1/20 0.36
JAK2 O60674 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
PAK4 O96013 1/20 0.36
CSF1R P07333 1/20 0.36
RET P07949 1/20 0.36
IGF1R P08069 1/20 0.36
FGFR1 P11362 1/20 0.36
PRKACA P17612 1/20 0.36
FLT1 P17948 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29680885 1.00 CYP2A6 (0.39) CYP2A6CDK8CYP1A2CYP3A4CYP2C8
SCHEMBL4171887 0.83 TGFBR1 (0.51) CDK8CYP3A4CYP2C8TGFBR1JAK1
SCHEMBL858844 0.77 IKBKB (0.64) CDK8IKBKBCHUKDAPK3JAK2
SCHEMBL4153879 0.75 TGFBR1 (0.47) CYP2A6CDK8CYP3A4CYP2C8TGFBR1
SCHEMBL29953681 0.73 CDK8 (0.50) CDK8JAK1IKBKBCHUKDAPK3
SCHEMBL29956462 0.73 MAPK1 (0.42) CDK8IKBKBCHUKDAPK3JAK2
SCHEMBL4157147 0.72 TGFBR1 (0.50) CYP2A6CDK8CYP3A4CYP2C8TGFBR1
SCHEMBL29681139 0.72 IKBKB (0.45) CYP2A6CDK8JAK1IKBKBCHUK
SCHEMBL24528672 0.72 IKBKB (0.45) CYP2A6CDK8JAK1IKBKBCHUK
SCHEMBL24528665 0.71 NEK1 (0.36) JAK1IKBKBCHUKALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed