SCHEMBL24528635

SCHEMBL24528635

CN(C)CCC/N=C/c1ccc(-c2nc(Cl)nc3[nH]ccc23)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BPTF Q12830 2/20 0.38
PDK1 Q15118 6/20 0.37
IKBKB O14920 2/20 0.33
CHUK O15111 2/20 0.33
JAK1 P23458 2/20 0.32
PDK2 Q15119 1/20 0.32
PDK3 Q15120 1/20 0.32
PDK4 Q16654 1/20 0.32
KDM4E B2RXH2 1/20 0.31
EGFR P00533 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
GABARAP O95166 1/20 0.31
GABARAPL2 P60520 1/20 0.31
MAP1LC3C Q9BXW4 1/20 0.31
MAP1LC3B Q9GZQ8 1/20 0.31
GABARAPL1 Q9H0R8 1/20 0.31
MAP1LC3A Q9H492 1/20 0.31
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29681028 1.00 BPTF (0.38) BPTFPDK1IKBKBCHUKJAK1
SCHEMBL24528663 0.81 KDM4E (0.39) PDK1IKBKBCHUKPDK2PDK3
SCHEMBL29680615 0.81 KDM4E (0.39) PDK1IKBKBCHUKPDK2PDK3
SCHEMBL29680982 0.77 NEK1 (0.36) BPTFIKBKBCHUKJAK1ALDH1A1
SCHEMBL24528665 0.77 NEK1 (0.36) BPTFIKBKBCHUKJAK1ALDH1A1
SCHEMBL29680804 0.76 TERT (0.41) BPTFPDK1LMNA
SCHEMBL24528583 0.74 KDM4E (0.38) KDM4EALDH1A1LMNA
SCHEMBL29680660 0.74 KDM4E (0.38) KDM4EALDH1A1LMNA
SCHEMBL24528672 0.72 IKBKB (0.45) PDK1IKBKBCHUKJAK1PDK2
SCHEMBL29681139 0.72 IKBKB (0.45) PDK1IKBKBCHUKJAK1PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed