SCHEMBL29680982

SCHEMBL29680982

CN(C)CCCCN=Cc1ccc(-c2cc(-c3ccc(C=NCCCCN(C)C)cc3)c3cc[nH]c3n2)cc1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NEK1 Q96PY6 2/20 0.36
IKBKB O14920 2/20 0.36
CHUK O15111 1/20 0.36
JAK1 P23458 10/20 0.35
BPTF Q12830 2/20 0.35
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
RIPK1 Q13546 1/20 0.32
PIM1 P11309 1/20 0.31
PIM3 Q86V86 1/20 0.31
HPGDS O60760 1/20 0.31
SYK P43405 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24528665 1.00 NEK1 (0.36) NEK1IKBKBCHUKJAK1BPTF
SCHEMBL29681210 0.81 JAK1 (0.39) IKBKBCHUKJAK1ALDH1A1SYK
SCHEMBL24528644 0.81 JAK1 (0.39) IKBKBCHUKJAK1ALDH1A1SYK
SCHEMBL29681028 0.77 BPTF (0.38) NEK1IKBKBCHUKJAK1BPTF
SCHEMBL24528635 0.77 BPTF (0.38) NEK1IKBKBCHUKJAK1BPTF
SCHEMBL29680686 0.76 TERT (0.41) NEK1IKBKBCHUKJAK1BPTF
SCHEMBL24528696 0.73 KDM4E (0.41) ALDH1A1LMNA
SCHEMBL29680758 0.73 KDM4E (0.41) ALDH1A1LMNA
Oxalic Acid SCHEMBL29680687 0.71 JAK1 (0.43) NEK1IKBKBCHUKJAK1
SCHEMBL24528632 0.71 CYP2A6 (0.39) IKBKBCHUKJAK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4263539-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE - INSERM (FR) 2023-10-25 EP disclosed
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed