SCHEMBL24528682

SCHEMBL24528682

O=Cc1ccc(-c2cc(-c3ccc(C=O)cc3)c3ccn(C=O)c3n2)cc1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
CYP11B1 P15538 1/20 0.33
CYP2A6 P11509 2/20 0.33
CDC7 O00311 1/20 0.32
PIM1 P11309 1/20 0.32
GSK3B P49841 1/20 0.32
HIPK2 Q9H2X6 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
DRD1 P21728 3/20 0.31
BRAF P15056 1/20 0.30
DRD2 P14416 1/20 0.30
DRD4 P21917 1/20 0.30
DRD5 P21918 1/20 0.30
DRD3 P35462 1/20 0.30
PTGS1 P23219 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29680818 0.76 ADORA2A (0.46) ALDH1A1MAPTCYP11B1
SCHEMBL24528641 0.76 ADORA2A (0.46) ALDH1A1MAPTCYP11B1
SCHEMBL29680970 0.73 HSP90AA1 (0.36) ALDH1A1MAPT
SCHEMBL24528676 0.73 HSP90AA1 (0.36) ALDH1A1MAPT
SCHEMBL29680885 0.68 CYP2A6 (0.39) ALDH1A1MAPTCYP2A6CLK4
SCHEMBL24528632 0.68 CYP2A6 (0.39) ALDH1A1MAPTCYP2A6CLK4
SCHEMBL26091984 0.67 ALDH1A1 (0.57) ALDH1A1MAPTCYP2A6BRAF
SCHEMBL23637796 0.67 ALDH1A1 (0.45) ALDH1A1MAPTCYP2A6DRD1BRAF
SCHEMBL24528698 0.66 ALDH1A1 (0.37) ALDH1A1MAPTDRD1DRD2DRD4
SCHEMBL6919033 0.64 CYP2A6 (0.48) ALDH1A1CYP2A6DRD1DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022129376-A1 6-6 OR 5-6 FUSED BICYCLIC COMPOUNDS COMPRISING A PYRI(MI)DINE RING USEFUL IN THE|TREATMENT OF INFECTIOUS DISEASES INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2022-06-23 WO disclosed