SCHEMBL2454397

SCHEMBL2454397

COC(=O)C(Cc1ccccc1)NC(=S)NCC1(C(C)(C)C)CCCN1C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
LMNA P02545 2/20 0.51
GLA P06280 1/20 0.51
ATM Q13315 3/20 0.49
POLB P06746 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
GFER P55789 1/20 0.46
GAA P10253 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
THRB P10828 1/20 0.43
HSD17B10 Q99714 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
NLRP3 Q96P20 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2454395 1.00 ALDH1A1 (0.51) ALDH1A1LMNAGLAATMPOLB
SCHEMBL2454516 0.85 MEN1 (0.37) ALDH1A1LMNAATMCYP2C9CYP2C19
SCHEMBL2489651 0.85 MEN1 (0.37) ALDH1A1LMNAATMCYP2C9CYP2C19
SCHEMBL2452733 0.81
SCHEMBL336767 0.78 LMNA (0.45) LMNA
SCHEMBL337364 0.78 LMNA (0.45) LMNA
SCHEMBL2454396 0.71 ATM (0.55) ALDH1A1LMNAGLAATMPOLB
SCHEMBL7983508 0.71 DPP7 (0.40) KMT2A
SCHEMBL20335018 0.70 ALDH1A1 (0.68) ALDH1A1LMNAGLAATMPOLB
SCHEMBL20335019 0.70 ALDH1A1 (0.68) ALDH1A1LMNAGLAATMPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2366700-A1 Pyrrolidine-thioxopyrimidinone/thiohydantoin organocatolysts National and Kapodistrian Universty of Athens (GR) 2011-09-21 EP disclosed