SCHEMBL24548682

SCHEMBL24548682

Cc1c(Oc2ccc(-n3nc(C#N)c(=O)[nH]c3=O)cc2F)n[nH]c(=O)c1C

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
THRA P10827 15/20 0.45
THRB P10828 15/20 0.45
CYP2C8 P10632 1/20 0.45
CYP2C9 P11712 1/20 0.45
MET P08581 3/20 0.32
ERBB2 P04626 1/20 0.32
F10 P00742 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24548665 0.88 THRA (0.45) THRATHRBCYP2C8CYP2C9
SCHEMBL25673742 0.88 THRA (0.54) THRATHRBCYP2C8CYP2C9
SCHEMBL25673739 0.84 THRA (0.58) THRATHRBCYP2C8CYP2C9
SCHEMBL25240420 0.81 THRA (0.49) THRATHRBCYP2C8CYP2C9
SCHEMBL24548722 0.81 THRA (0.67) THRATHRBCYP2C8CYP2C9
SCHEMBL22660393 0.80 THRA (0.66) THRATHRBCYP2C8CYP2C9
SCHEMBL24548661 0.77 THRA (0.45) THRATHRBCYP2C8CYP2C9
SCHEMBL24548673 0.75 THRA (0.43) THRATHRBCYP2C8CYP2C9
SCHEMBL23245118 0.70 THRA (0.68) THRATHRBCYP2C8CYP2C9
SCHEMBL23245106 0.70 THRA (0.68) THRATHRBCYP2C8CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022127779-A1 SUBSTITUTED PYRIDAZINONE COMPOUND AND USE THEREOF 山东第一医科大学(山东省医学科学院) 2022-06-23 WO disclosed