SCHEMBL24554356

SCHEMBL24554356

Nc1ccc(C#Cc2ccccc2F)cc1F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 4/20 0.53
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C9 P11712 1/20 0.44
HPGD P15428 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
GFER P55789 1/20 0.43
FFAR1 O14842 6/20 0.42
FFAR4 Q5NUL3 5/20 0.42
CASP3 P42574 1/20 0.41
SENP8 Q96LD8 1/20 0.41
SENP7 Q9BQF6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3708035 0.83 MAPT (0.54) GRM5ALDH1A1KDM4EMEN1NPC1
SCHEMBL24294400 0.81 CYP11B1 (0.43) GRM5ALDH1A1KDM4EMEN1NPC1
SCHEMBL27682554 0.77 APP (0.58) GRM5ALDH1A1MEN1NPC1MAPT
SCHEMBL5401212 0.77 APP (0.55) GRM5ALDH1A1KDM4EMEN1NPC1
SCHEMBL30270412 0.77 CYP3A4 (0.59) GRM5ALDH1A1KDM4EMEN1NPC1
SCHEMBL10300113 0.76 GRM5 (0.54) GRM5CYP1A2GFERFFAR1FFAR4
SCHEMBL29251289 0.76 GRM5 (0.52) GRM5ALDH1A1KDM4EMEN1NPC1
SCHEMBL9305673 0.75 GRM5 (0.51) GRM5ALDH1A1KDM4EMEN1NPC1
SCHEMBL30270426 0.75 KDM4E (0.53) GRM5ALDH1A1KDM4EMEN1NPC1
SCHEMBL8424794 0.74 APP (0.57) GRM5ALDH1A1KDM4EMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022128845-A1 HETEROAROMATIC ISOTHIOCYANATES MERCK PATENT GMBH (DE) 2022-06-23 WO disclosed