SCHEMBL24558265

SCHEMBL24558265

Cn1cnc2c(Br)c(Cl)c(F)c(C(=O)O)c21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A2 P19784 5/20 0.35
CSNK2A1 P68400 4/20 0.35
NR3C1 P04150 2/20 0.33
KDM4C Q9H3R0 2/20 0.32
KDM2B Q8NHM5 1/20 0.32
CSNK2B P67870 2/20 0.31
CSNK2A3 Q8NEV1 2/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
EGLN1 Q9GZT9 1/20 0.30
SMC2 O95347 1/20 0.30
EGFR P00533 1/20 0.30
MAP2K2 P36507 1/20 0.30
MAP2K1 Q02750 1/20 0.30
SMC1A Q14683 1/20 0.30
AAK1 Q2M2I8 1/20 0.30
Q6ZSR9 Q6ZSR9 1/20 0.30
BMP2K Q9NSY1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL615255 0.81 NR3C1 (0.33) NR3C1KDM4CPDE4APDE4BPDE4C
SCHEMBL31107272 0.72 DPP4 (0.39) KDM4CKDM2B
SCHEMBL24558219 0.72 HTT (0.33) NR3C1
SCHEMBL24558204 0.69 ADORA2A (0.32)
SCHEMBL1343248 0.66 CDK1 (0.42) NR3C1KDM4CKDM2B
SCHEMBL4323205 0.66 MAPK14 (0.37) KDM4CKDM2BPDE4APDE4BPDE4C
SCHEMBL616982 0.65 MAP2K2 (0.37) CSNK2A2KDM4CKDM2BEGLN1SMC2
SCHEMBL21068031 0.64 CSNK2A1 (0.52) CSNK2A2CSNK2A1CSNK2BCSNK2A3
SCHEMBL11633469 0.64 CDK1 (0.43) NR3C1
SCHEMBL10290716 0.63 CDK1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3935060-B1 FUSED TRICYCLIC COMPOUNDS USEFUL AS ANTICANCER AGENTS ASTRAZENECA AB (SE) 2023-11-15 EP disclosed
US-20220204527-A1 FUSED TRICYCLIC COMPOUNDS USEFUL AS ANTICANCER AGENTS ASTRAZENECA UK LIMITED (GB) 2022-06-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220204527-A1 FUSED TRICYCLIC COMPOUNDS USEFUL AS ANTICANCER AGENTS MCL1, TP53, CCNA2 CSNK2A2 865/4885CSNK2A1 902/4885NR3C1 3466/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.