SCHEMBL2456152

SCHEMBL2456152

Cn1nc(-c2nc(-c3ccc(N4CCC(O)CC4)cc3)no2)c2c1CC(C)(C)CC2

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 4/20 0.33
S1PR3 Q99500 1/20 0.33
MAPT P10636 1/20 0.32
DGAT1 O75907 3/20 0.31
BCL2L1 Q07817 1/20 0.31
ALOX5AP P20292 1/20 0.31
CHEK1 O14757 1/20 0.31
HIF1A Q16665 1/20 0.31
PIK3CA P42336 1/20 0.31
MTOR P42345 1/20 0.31
CFTR P13569 1/20 0.30
HDAC4 P56524 1/20 0.30
BCL2 P10415 1/20 0.30
TP53 P04637 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2473284 0.81 S1PR1 (0.40) S1PR1S1PR3MAPTTP53
SCHEMBL2472405 0.81 RARA (0.40) S1PR1S1PR3MAPT
SCHEMBL2456203 0.79 S1PR1 (0.44) S1PR1S1PR3
SCHEMBL2470344 0.78 CA9 (0.48) S1PR1
SCHEMBL2476438 0.76 MAPK1 (0.39) S1PR1S1PR3MAPT
SCHEMBL2473364 0.76 MAPT (0.42) S1PR1MAPTTP53
SCHEMBL2472532 0.76 CDK4 (0.36) S1PR1MAPTALOX5APPIK3CAMTOR
SCHEMBL2474719 0.75 DGAT1 (0.39) S1PR1S1PR3MAPTDGAT1BCL2L1
SCHEMBL2467513 0.74 S1PR1 (0.38) S1PR1S1PR3MAPT
SCHEMBL2470317 0.74 BCL2L1 (0.37) S1PR1S1PR3MAPTDGAT1BCL2L1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011113578-A1 NEW OXADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2011-09-22 WO claimed
EP-2366702-A1 New oxadiazole derivatives Almirall, S.A. (ES) 2011-09-21 EP claimed
WO-2011113578-A1 NEW OXADIAZOLE DERIVATIVES ALMIRALL, S.A. (ES) 2011-09-22 WO disclosed
EP-2366702-A1 New oxadiazole derivatives Almirall, S.A. (ES) 2011-09-21 EP disclosed
EP-2366702-A1 New oxadiazole derivatives Almirall, S.A. (ES) 2011-09-21 EP disclosed