SCHEMBL2456582

SCHEMBL2456582

COc1ccc(-n2ncc(C)c2C(=O)O)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.51
NPC1 O15118 3/20 0.51
RAB9A P51151 3/20 0.51
MAPT P10636 2/20 0.51
NFKB1 P19838 1/20 0.51
NFKB2 Q00653 1/20 0.51
RELA Q04206 1/20 0.51
MAPK14 Q16539 1/20 0.50
PTPN1 P18031 1/20 0.49
NPBWR1 P48145 6/20 0.48
MCHR1 Q99705 4/20 0.48
PKM P14618 1/20 0.48
HTT P42858 2/20 0.48
S1PR4 O95977 1/20 0.48
ALDH1A1 P00352 1/20 0.48
S1PR1 P21453 1/20 0.48
KMT2A Q03164 1/20 0.48
PAX8 Q06710 1/20 0.48
TP53 P04637 1/20 0.47
MAPKAPK2 P49137 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4300658 0.82 MAPK1 (0.54) SMN1; SMN2NPC1RAB9AMAPTPKM
SCHEMBL5788758 0.80 HTT (0.48) SMN1; SMN2NPC1RAB9AMAPTNFKB1
SCHEMBL2855932 0.79 NPC1 (0.69) SMN1; SMN2NPC1RAB9AMAPTNFKB1
SCHEMBL16060701 0.78 XDH (0.45) NPC1RAB9AMAPK14RPA1
SCHEMBL12991623 0.77 NPC1 (0.51) SMN1; SMN2NPC1RAB9AMAPTNFKB1
SCHEMBL15897901 0.76 SMN1; SMN2 (0.50) SMN1; SMN2NPC1RAB9AMAPTHTT
SCHEMBL16252260 0.75 UCHL1 (0.54) MAPTNPBWR1MCHR1ALDH1A1
SCHEMBL3296237 0.75 PTPN1 (0.79) SMN1; SMN2NPC1RAB9AMAPTNFKB1
SCHEMBL10365375 0.75 PTPN1 (0.57) SMN1; SMN2NPC1RAB9AMAPTNFKB1
SCHEMBL460952 0.74 MAPK14 (0.54) MAPK14ALDH1A1KMT2ATP53HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1988777-B1 PYRAZOLES FOR THE TREATMENT OF OBESITY AND OTHER CNS DISORDERS ATHERSYS INC (US) 2011-09-21 EP disclosed