SCHEMBL2456751

SCHEMBL2456751

Cc1cnc(C(=O)NC2Cc3ccsc3C2)c(N)n1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 11/20 0.39
ACVR2A P27037 1/20 0.39
TGFBR2 P37173 1/20 0.39
SCN4A P35499 1/20 0.36
SCN3A Q9NY46 1/20 0.36
GRM5 P41594 2/20 0.36
ACVR1 Q04771 2/20 0.35
ATR Q13535 1/20 0.34
ADORA2A P29274 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2456743 0.83 PRKCI (0.42) CHRM4GRM5ATR
SCHEMBL2458764 0.77 HDAC1 (0.48) GRM5KDM4EALDH1A1
SCHEMBL2459809 0.77 RAB9A (0.40) CHRM4ADORA2AALDH1A1
SCHEMBL2456197 0.74 PRKCI (0.45) CHRM4KDM4EALDH1A1
Trifluoroacetic Acid SCHEMBL27607866 0.73 KMT2A (0.43) GRM5KDM4E
SCHEMBL2454980 0.73 EGFR (0.42) CHRM4ADORA2A
SCHEMBL2454948 0.72 CNR1 (0.48) CHRM4ALDH1A1
Trifluoroacetic Acid SCHEMBL27626866 0.70 PRKCI (0.42) CHRM4KDM4EALDH1A1
SCHEMBL2456714 0.70 GPR183 (0.46) ADORA2A
SCHEMBL2454974 0.68 NPC1 (0.43) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534277-B1 ACYLATED, HETEROARYL-CONDENSED CYCLOALKENYLAMINES AND THEIR USE AS PHARMACEUTICALS SANOFI AVENTIS DEUTSCHLAND (DE) 2011-09-14 EP disclosed
EP-1534277-B1 ACYLATED, HETEROARYL-CONDENSED CYCLOALKENYLAMINES AND THEIR USE AS PHARMACEUTICALS SANOFI AVENTIS DEUTSCHLAND (DE) 2011-09-14 EP disclosed