SCHEMBL24568601

SCHEMBL24568601

C=C(C)[C@@H](C)NC(=O)OCC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.39
LMNA P02545 1/20 0.39
CYP3A4 P08684 1/20 0.39
NFKB1 P19838 1/20 0.39
ADRA1A P35348 1/20 0.39
RAB9A P51151 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
KMT2A Q03164 1/20 0.39
CTSK P43235 1/20 0.37
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA7 P43166 1/20 0.31
FSHR P23945 1/20 0.30
TPSAB1 Q15661 2/20 0.30
PLG P00747 1/20 0.30
PRSS1 P07477 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13127979 0.85 TSHR (0.41) TSHRLMNACYP3A4NFKB1ADRA1A
SCHEMBL22649551 0.81 TYR (0.41) TSHRLMNACYP3A4NFKB1ADRA1A
SCHEMBL12890775 0.79 TSHR (0.56) TSHRLMNACYP3A4NFKB1ADRA1A
SCHEMBL29068653 0.76 CA1 (0.49) TSHRLMNAKMT2ACTSKCA1
SCHEMBL24427421 0.76 HRH3 (0.43) TSHRLMNACYP3A4NFKB1ADRA1A
SCHEMBL24567503 0.76 TSHR (0.41) TSHRLMNACYP3A4NFKB1ADRA1A
SCHEMBL16181347 0.75 TSHR (0.33) TSHR
SCHEMBL68958 0.73 TSHR (0.43) TSHRLMNACYP3A4NFKB1ADRA1A
SCHEMBL20854165 0.71 CA1 (0.49) KMT2ACTSKCA1CA2CA7
SCHEMBL20854166 0.71 CA1 (0.49) KMT2ACTSKCA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022140428-A2 INHIBITORS OF PEPTIDYLARGININE DEIMINASES GILEAD SCIENCES, INC. (US) 2022-06-30 WO disclosed