SCHEMBL24570925

SCHEMBL24570925

Cc1cc(C)c(-c2ccccc2)c(N)c1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.44
AKT2 P31751 2/20 0.44
TDO2 P48775 1/20 0.44
KMT2A Q03164 1/20 0.44
MAPT P10636 2/20 0.42
CYP3A4 P08684 3/20 0.42
TDP1 Q9NUW8 3/20 0.42
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
CDK8 P49336 1/20 0.42
ACVR1 Q04771 1/20 0.42
PTPN1 P18031 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
TSHR P16473 1/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3974332 0.85 AKT2 (0.48) BRD4AKT2TDO2KMT2AMAPT
SCHEMBL27552263 0.83 TDP1 (0.41) BRD4AKT2TDO2KMT2AMAPT
SCHEMBL16429717 0.81 RPS6KA3 (0.47) BRD4AKT2TDO2KMT2AMAPT
SCHEMBL28060692 0.80 KMT2A (0.40) BRD4AKT2TDO2KMT2AMAPT
SCHEMBL5551256 0.80 MAPT (0.42) BRD4AKT2KMT2AMAPTSMN1; SMN2
SCHEMBL3794847 0.79 CYP3A4 (0.46) BRD4AKT2TDO2KMT2AMAPT
SCHEMBL3145455 0.79 MAPT (0.42) BRD4AKT2KMT2AMAPTCDK8
SCHEMBL675595 0.79 ALDH1A1 (0.50) BRD4AKT2TDO2KMT2AMAPT
SCHEMBL28535205 0.79 ALDH1A1 (0.50) BRD4AKT2TDO2KMT2AMAPT
SCHEMBL26782066 0.79 ESR2 (0.41) BRD4AKT2TDO2KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4019520-A1 HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE INCLUDING HETEROCYCLIC COMPOUND, AND ELECTRONIC APPARATUS INCLUDING ORGANIC LIGHT-EMITTING DEVICE Samsung Electronics Co., Ltd. (KR) 2022-06-29 EP disclosed