SCHEMBL24574151

SCHEMBL24574151

CC(C)(O)c1cn2ccnc2cn1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.35
KEAP1 Q14145 1/20 0.35
NAMPT P43490 5/20 0.34
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
KMT2A Q03164 1/20 0.33
SSTR4 P31391 1/20 0.33
TGFBR1 P36897 4/20 0.32
MCHR1 Q99705 1/20 0.30
MET P08581 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10183355 0.85 DYRK1A (0.37) DYRK1AKEAP1NAMPTMEN1CYP1A2
SCHEMBL24574341 0.83 NAMPT (0.34) DYRK1AKEAP1NAMPTMEN1CYP1A2
SCHEMBL19969731 0.79 KEAP1 (0.37) DYRK1AKEAP1NAMPTMEN1CYP1A2
SCHEMBL29837274 0.78 NAMPT (0.40) DYRK1AKEAP1NAMPTMEN1CYP1A2
SCHEMBL19969788 0.77 KEAP1 (0.35) DYRK1AKEAP1NAMPTMEN1CYP1A2
SCHEMBL22726755 0.73 SSTR4 (0.33) SSTR4
SCHEMBL2629380 0.72 TGFBR1 (0.43) DYRK1AKEAP1NAMPTMEN1CYP1A2
Trifluoroacetic Acid SCHEMBL30804022 0.72 NAMPT (0.42) NAMPTMEN1CYP1A2KMT2AMCHR1
SCHEMBL19950935 0.71 SSTR4 (0.49) DYRK1AKEAP1MEN1CYP1A2KMT2A
SCHEMBL5487376 0.71 DYRK1A (0.40) DYRK1AKEAP1NAMPTMEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12612410-B2 Multi-cyclic IRAK and FLT3 inhibiting compounds and uses thereof CHILDREN'S HOSPITAL MEDICAL CENTER (US) 2026-04-28 US disclosed
WO-2023250431-A9 MULTI-CYCLIC IRAK AND FLT3 INHIBITING COMPOUNDS AND USES THEREOF CHILDREN'S HOSPITAL MEDICAL CENTER (US) 2025-03-06 WO disclosed
US-20240294530-A1 MULTI-CYCLIC IRAK AND FLT3 INHIBITING COMPOUNDS AND USES THEREOF CHILDREN'S HOSPITAL MEDICAL CENTER 2024-09-05 US disclosed
WO-2022140647-A1 MULTI-CYCLIC IRAK AND FLT3 INHIBITING COMPOUNDS AND USES THEREOF CHILDREN'S HOSPITAL MEDICAL CENTER (US) 2022-06-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240294530-A1 MULTI-CYCLIC IRAK AND FLT3 INHIBITING COMPOUNDS AND USES THEREOF FLT3, IRAK1, IRAK2 DYRK1A 631/4885KEAP1 1161/4885NAMPT 2457/4885
US-12612410-B2 Multi-cyclic IRAK and FLT3 inhibiting compounds and uses thereof FLT3, IRAK3, IRAK2 DYRK1A 1980/4885KEAP1 1096/4885NAMPT 3706/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.