SCHEMBL24575646

SCHEMBL24575646

Oc1cc(C(F)(F)F)ccc1-c1nnc(N[C@@H]2CCCNC2)c2c1COCC2

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 7/20 0.59
IL1B P01584 7/20 0.50
CHEK2 O96017 4/20 0.46
CHEK1 O14757 2/20 0.46
KCNH2 Q12809 1/20 0.44
IDH2 P48735 1/20 0.41
IRAK4 Q9NWZ3 1/20 0.40
PDPK1 O15530 1/20 0.40
RPS6KB1 P23443 1/20 0.40
PIM1 P11309 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24575648 0.96 NLRP3 (0.59) NLRP3IL1BCHEK2CHEK1KCNH2
SCHEMBL24575703 0.93 NLRP3 (0.68) NLRP3IL1BCHEK2CHEK1KCNH2
SCHEMBL31057145 0.93 NLRP3 (0.68) NLRP3IL1BCHEK2CHEK1KCNH2
Hydrochloric Acid SCHEMBL31057406 0.92 NLRP3 (0.67) NLRP3IL1BCHEK2CHEK1KCNH2
SCHEMBL24575084 0.90 IL1B (0.56) NLRP3IL1BCHEK2CHEK1KCNH2
SCHEMBL31057311 0.90 NLRP3 (0.57) NLRP3IL1BCHEK2CHEK1KCNH2
SCHEMBL28934266 0.90 IL1B (0.56) NLRP3IL1BCHEK2CHEK1KCNH2
SCHEMBL30108758 0.90 IL1B (0.56) NLRP3IL1BCHEK2CHEK1KCNH2
SCHEMBL30214109 0.89 IL1B (0.55) NLRP3IL1BCHEK2CHEK1KCNH2
SCHEMBL29275600 0.89 IL1B (0.55) NLRP3IL1BCHEK2CHEK1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022135567-A1 PYRIDAZINE-CONTAINING COMPOUND AND MEDICINAL USE THEREOF 上海拓界生物医药科技有限公司 2022-06-30 WO disclosed