SCHEMBL2460080

SCHEMBL2460080

CCN(CC)c1[c]c2ccccc2cc1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 1/20 0.33
TSHR P16473 1/20 0.33
ELANE P08246 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TERT O14746 1/20 0.32
CYP1A2 P05177 2/20 0.32
LMNA P02545 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
CYP2A6 P11509 1/20 0.31
BCHE P06276 2/20 0.31
ACHE P22303 2/20 0.31
MAPT P10636 1/20 0.31
CNR2 P34972 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720954 0.90 BCHE (0.30) TSHRBCHE
SCHEMBL2460446 0.87 ELANE (0.37) ELANELMNABCHEMAPT
SCHEMBL2462799 0.85 BCHE (0.31) BCHEMAPT
SCHEMBL2459368 0.84 KCNH2 (0.38) ELANECYP1A2LMNACYP2D6CYP2C19
SCHEMBL2456300 0.83 CYP1A2 (0.31) CYP1A2CYP2A6
SCHEMBL2459934 0.82 ELANE (0.38) ELANELMNABCHEMAPT
SCHEMBL2456814 0.81 ELANE (0.35) ELANECYP1A2LMNACYP2D6CYP2C19
SCHEMBL4722542 0.80 ELANE (0.37) ELANELMNABCHEMAPT
SCHEMBL2456330 0.80 KCNH2 (0.36) ELANECYP1A2LMNACYP2D6CYP2C19
SCHEMBL6553704 0.78 TSHR (0.39) TSHRCYP2C19ACHECNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 48 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040116703-A1 8-Azabicyclo[3.2.1]oct-2-ene and -octane derivatives technical field NEUROSEARCH A/S 2004-06-17 US claimed
EP-1133494-B1 8-AZABICYCLO 3.2.1]OCT-2-ENE AND -OCTANE DERIVATIVES NEUROSEARCH AS (DK) 2004-02-18 EP claimed
US-6680328-B2 CHOLINERGIC LIGANDS OF NICOTINIC ACETYL CHOLINE RECEPTORS FOR TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, SMOOTH MUSCLE CONTRACTION DISORDERS, ENDOCRINE DISEASES/DISORDERS, NEURODEGENERATION, INFLAMMATION, PAIN, AND DRUG WITHDRAWAL NEUROSEARCH A/S (DK) 2004-01-20 US claimed
US-20020035122-A1 8-azabicyclo[3.2.1]oct-2-ene and -octane derivatives ANIONA APS (DK) 2002-03-21 US claimed
EP-1133494-A1 8-AZABICYCLO 3.2.1]OCT-2-ENE AND -OCTANE DERIVATIVES NEUROSEARCH A/S (DK) 2001-09-19 EP claimed
WO-2000032600-A1 8-AZABICYCLO[3.2.1]OCT-2-ENE AND -OCTANE DERIVATIVES NEUROSEARCH A/S (DK) 2000-06-08 WO claimed
EP-2524686-B1 PIGMENTATION-PREVENTING OR -AMELIORATING AGENT POLA CHEM IND INC (JP) 2017-06-21 EP disclosed
EP-2514402-B1 PREVENTING OR AMELIORATING AGENT FOR PIGMENTATION POLA CHEM IND INC (JP) 2016-08-31 EP disclosed
US-9414998-B2 Preventing or ameliorating agent for pigmentation POLA CHEMICAL INDUSTRIES INC. (JP) 2016-08-16 US disclosed
US-9066914-B2 Prophylactic or ameliorating agent for pigmentation POLA CHEMICAL INDUSTRIES INC. (JP) 2015-06-30 US disclosed
US-20140322150-A1 PREVENTING OR AMELIORATING AGENT FOR PIGMENTATION POLA CHEMICAL INDUSTRIES INC. (JP) 2014-10-30 US disclosed
EP-2524686-A1 PIGMENTATION-PREVENTING OR -AMELIORATING AGENT Pola Chemical Industries Inc. (JP) 2012-11-21 EP disclosed
US-20120282203-A1 PROPHYLACTIC OR AMELIORATING AGENT FOR PIGMENTATION POLA CHEMICAL INDUSTRIES INC. (JP) 2012-11-08 US disclosed
US-5035969-A And a compound in a photoconductive layer on a support; high potential stability, durability FUJI PHOTO FILM CO., LTD. (JP) 1991-07-30 US disclosed
US-4985323-A Photoconductor, Sensitizer, Amide FUJI PHOTO FILM CO., LTD. (JP) 1991-01-15 US disclosed
US-4943681-A PHTHALOCYANINE COMPLEX, HIGH SENSITIVITY, LASERS TOYO INK MANUFACTURING CO., LTD. (JP) 1990-07-24 US disclosed
EP-0376745-A2 Optical recording medium and process for the production thereof TOYO INK MANUFACTURING CO., LTD. (JP) 1990-07-04 EP disclosed
US-4411812-A Dichroic liquid crystal compositions made with asymmetric tris-azo dyes GENERAL ELECTRIC COMPANY (US) 1983-10-25 US disclosed
US-4411812-A Dichroic liquid crystal compositions made with asymmetric tris-azo dyes GENERAL ELECTRIC COMPANY (US) 1983-10-25 US disclosed
US-4256458-A DIMERIC PYRIDINIUM DYES BASF AKTIENGESELLSCHAFT (DE) 1981-03-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020035122-A1 8-azabicyclo[3.2.1]oct-2-ene and -octane derivatives CHRNA2, CHRNA7, CHRNA10 ACP1 4220/4885TSHR 216/4885ELANE 1312/4885
US-20120282203-A1 PROPHYLACTIC OR AMELIORATING AGENT FOR PIGMENTATION TYR, MC1R, NQO1 ACP1 2998/4885TSHR 2578/4885ELANE 691/4885
US-20140322150-A1 PREVENTING OR AMELIORATING AGENT FOR PIGMENTATION TYR, MC1R, MITF ACP1 2054/4885TSHR 1691/4885ELANE 535/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.