SCHEMBL24601240

SCHEMBL24601240

C=CNC(=O)[C@@H]1C[C@@H](O)[C@H](n2cnc3c(NCc4ccccn4)nc(-c4cncc(Cl)c4)nc32)O1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NT5E P21589 1/20 0.42
ADORA3 P0DMS8 11/20 0.39
ADORA2A P29274 4/20 0.36
ADORA1 P30542 3/20 0.36
KCNA5 P22460 1/20 0.36
KCNH2 Q12809 1/20 0.36
ADORA2B P29275 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24600684 0.92 NT5E (0.40) NT5EADORA3ADORA2AADORA1KCNA5
SCHEMBL24601100 0.92 NT5E (0.40) NT5EADORA3ADORA2AADORA1KCNA5
SCHEMBL24600671 0.91 ADORA3 (0.45) NT5EADORA3ADORA2AADORA1ADORA2B
SCHEMBL24601006 0.91 ADORA3 (0.48) NT5EADORA3ADORA2AADORA1ADORA2B
SCHEMBL24600934 0.90 KCNA5 (0.44) NT5EADORA3ADORA2AADORA1KCNA5
SCHEMBL24601230 0.90 NT5E (0.43) NT5EADORA3ADORA2AADORA1KCNA5
SCHEMBL24601226 0.90 ADORA3 (0.44) NT5EADORA3ADORA2AADORA1ADORA2B
SCHEMBL24601231 0.90 NT5E (0.42) NT5EADORA3ADORA2AADORA1KCNA5
SCHEMBL24601184 0.89 ADORA3 (0.38) NT5EADORA3ADORA2AADORA1ADORA2B
SCHEMBL24601238 0.88 NT5E (0.42) NT5EADORA3ADORA2AADORA1KCNA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022143740-A1 ADENOSINE A3 RECEPTOR AGONIST, PREPARATION METHOD THEREFOR, AND USE THEREOF 浙江春禾医药科技有限公司 2022-07-07 WO disclosed