SCHEMBL24601279

SCHEMBL24601279

CNC(=O)[C@@H]1C[C@@H](O)[C@H](n2cnc3c(NCc4cccc(Cl)n4)nc(-c4cncc(Cl)c4)nc32)O1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 11/20 0.50
ADORA2A P29274 4/20 0.45
ADORA1 P30542 4/20 0.45
ADORA2B P29275 2/20 0.45
MAPK1 P28482 3/20 0.44
TP53 P04637 2/20 0.44
MAPT P10636 2/20 0.44
HTR2C P28335 1/20 0.44
PPARG P37231 1/20 0.44
HTR2B P41595 1/20 0.44
PPARD Q03181 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.44
CYP1A2 P05177 1/20 0.44
NPC1 O15118 1/20 0.41
GMNN O75496 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
THRB P10828 1/20 0.41
HPGD P15428 1/20 0.41
BLM P54132 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24601006 0.92 ADORA3 (0.48) ADORA3ADORA2AADORA1ADORA2BMAPK1
SCHEMBL24600970 0.92 ADORA3 (0.47) ADORA3ADORA2AADORA1ADORA2BMAPK1
SCHEMBL24600751 0.89 ADORA3 (0.56) ADORA3ADORA2AADORA1ADORA2BMAPK1
SCHEMBL24601019 0.88 ADORA3 (0.47) ADORA3ADORA2AADORA1ADORA2BMAPK1
SCHEMBL24601230 0.87 NT5E (0.43) ADORA3ADORA2AADORA1ADORA2BMAPK1
SCHEMBL24601571 0.87 ADORA3 (0.51) ADORA3ADORA2AADORA1ADORA2BMAPK1
SCHEMBL24601112 0.87 ADORA3 (0.44) ADORA3ADORA2AADORA1ADORA2BMAPK1
SCHEMBL24601231 0.86 NT5E (0.42) ADORA3ADORA2AADORA1ADORA2B
SCHEMBL24601226 0.86 ADORA3 (0.44) ADORA3ADORA2AADORA1ADORA2BTSHR
SCHEMBL24600931 0.86 ADORA3 (0.46) ADORA3ADORA2AADORA1ADORA2BMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022143740-A1 ADENOSINE A3 RECEPTOR AGONIST, PREPARATION METHOD THEREFOR, AND USE THEREOF 浙江春禾医药科技有限公司 2022-07-07 WO disclosed