SCHEMBL246068

SCHEMBL246068

COC(=O)c1ccc2ccccc2c1C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
KDM4E B2RXH2 3/20 0.51
ALDH1A1 P00352 3/20 0.51
NCEH1 Q6PIU2 2/20 0.51
HPGD P15428 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
HDAC3 O15379 1/20 0.49
HDAC4 P56524 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
HDAC9 Q9UKV0 1/20 0.49
HDAC5 Q9UQL6 1/20 0.49
SLC6A2 P23975 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6939268 0.87 NCEH1 (0.49) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL593520 0.84 MAPT (0.61) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL30356865 0.84 MAPT (0.61) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL13880496 0.83 CDC25B (0.63) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL71131 0.82 NCEH1 (0.59) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL8782101 0.82 MAPT (0.52) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL29404644 0.82 NCEH1 (0.59) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL244541 0.82 LDHA (0.62) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL161927 0.82 MAPT (0.52) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL16384835 0.81 MAPT (0.56) MAPTMEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120302722-A1 COPOLYETHER ESTER ELASTOMER INVISTA NORTH AMERICA S.A.R.L (US) 2012-11-29 US claimed
EP-2510039-A1 COPOLYETHER ESTER ELASTOMER Invista Technologies S.à.r.l. (CH) 2012-10-17 EP claimed
WO-2011071558-A1 COPOLYETHER ESTER ELASTOMER INVISTA TECHNOLOGIES S.A R.L. (CH) 2011-06-16 WO claimed
CN-118580225-A PRMT5-MTA synergistic inhibitor and application thereof 甘李药业股份有限公司 2024-09-03 CN disclosed
CN-111936576-B Thermoplastic resin composition and molded product made therefrom 乐天化学株式会社 2023-10-17 CN disclosed
CN-111936576-A Thermoplastic resin composition and molded product made therefrom 乐天化学株式会社 2020-11-13 CN disclosed
WO-2018005249-A1 BENZOISOQUINOLINONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK SHARP & DOHME CORP. (US) 2018-01-04 WO disclosed
WO-2017160670-A1 M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS AND METHODS OF USE THEREOF MERCK SHARP & DOHME CORP. (US) 2017-09-21 WO disclosed
WO-2017160670-A1 M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS AND METHODS OF USE THEREOF MERCK SHARP & DOHME CORP. (US) 2017-09-21 WO disclosed
EP-2709451-B1 N-LINKED LACTAM M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK SHARP & DOHME (US) 2015-12-30 EP disclosed
EP-2709451-B1 N-LINKED LACTAM M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK SHARP & DOHME (US) 2015-12-30 EP disclosed
WO-2010110554-A2 ORGANIC ELECTROLUMINESCENT DEVICE USING ORGANIC ELECTROLUMINESCENT COMPOUNDS DOW ADVANCED DISPLAY MATERIALS,LTD. (KR) 2010-09-30 WO disclosed
US-6833428-B1 Polyetherester elastomer ASAHI KASEI KABUSHIKI KAISHA (JP) 2004-12-21 US disclosed
US-5643925-A COGNITION ACTIVATORS AND NERVE GROWTH FACTORS SANKYO COMPANY, LIMITED (JP) 1997-07-01 US disclosed
US-5614521-A NERVE GROWTH FACTOR SANKYO COMPANY, LIMITED (JP) 1997-03-25 US disclosed
EP-0501656-B1 New benzene derivatives having (NGF) production-promoting activity SANKYO CO (JP) 1997-01-22 EP disclosed
EP-0501656-A2 New benzene derivatives having (NGF) production-promoting activity Sankyo Company Limited (JP) 1992-09-02 EP disclosed
US-4757130-A Condensation polymers with pendant side chains exhibiting nonlinear optical response HOECHST CELANESE CORPORATON (US) 1988-07-12 US disclosed
US-4540705-A Antidepressant imidazolines and related compounds STERLING DRUG INC. (US) 1985-09-10 US disclosed
EP-0125410-A2 Imidazolines and related compounds and preparation thereof STERLING DRUG INC. (US) 1984-11-21 EP disclosed