SCHEMBL2462007

SCHEMBL2462007

CN1CCC(NC(=O)O)C1=O

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.41
MAPK1 P28482 1/20 0.38
SCN9A Q15858 2/20 0.37
NAMPT P43490 1/20 0.36
APOL1 O14791 1/20 0.36
MME P08473 1/20 0.34
ACE P12821 1/20 0.34
FPR2 P25090 2/20 0.34
FPR1 P21462 1/20 0.34
NAAA Q02083 1/20 0.34
RIPK1 Q13546 5/20 0.34
DGAT2 Q96PD7 1/20 0.33
BRD4 O60885 1/20 0.33
TYK2 P29597 1/20 0.33
STAT3 P40763 1/20 0.33
MAP4K1 Q92918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6385322 1.00 HPGDS (0.41) HPGDSMAPK1SCN9ANAMPTAPOL1
SCHEMBL2464736 0.89 NAMPT (0.43) HPGDSMAPK1NAMPTMMEACE
SCHEMBL5639144 0.87 NAMPT (0.47) NAMPTMMEACENAAA
SCHEMBL15998895 0.85 HPGDS (0.41) HPGDSMAPK1SCN9ANAMPTAPOL1
SCHEMBL23022786 0.83 HPGDS (0.41) HPGDSMAPK1SCN9ANAMPTAPOL1
SCHEMBL30107181 0.83 HPGDS (0.41) HPGDSMAPK1SCN9ANAMPTAPOL1
SCHEMBL21246180 0.83 HPGDS (0.41) HPGDSMAPK1SCN9ANAMPTAPOL1
SCHEMBL27749158 0.83 HPGDS (0.36) HPGDSMAPK1SCN9ANAMPTAPOL1
SCHEMBL27283601 0.80 CYP1A2 (0.40) HPGDSSCN9ANAMPTMMEACE
SCHEMBL10713076 0.79 NAMPT (0.55) HPGDSNAMPTDGAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8026233-B2 P38 inhibitors and methods of use thereof ARRAY BIOPHARMA INC. (US) 2011-09-27 US disclosed
US-20090149443-A1 P38 INHIBITORS AND METHODS OF USE THEREOF ARRAY BIOPHARMA, INC. 2009-06-11 US disclosed
EP-1458684-A2 THERAPEUTIC HETEROCYCLES AstraZeneca AB (SE) 2004-09-22 EP disclosed
WO-2003051276-A2 THERAPEUTIC HETEROCYCLES ASTRAZENECA AB (SE) 2003-06-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090149443-A1 P38 INHIBITORS AND METHODS OF USE THEREOF MAPK1, MAPK4, BRIX1 HPGDS 2025/4885MAPK1 1/4885SCN9A 4411/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.