SCHEMBL24620294

SCHEMBL24620294

CCN(c1ccccc1)c1ccccn1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.55
CYP2C19 P33261 1/20 0.55
DHFR P00374 2/20 0.48
HCN1 O60741 2/20 0.46
HCN4 Q9Y3Q4 2/20 0.46
ALDH1A1 P00352 3/20 0.44
MAPT P10636 1/20 0.44
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CYP1A2 P05177 1/20 0.43
TSHR P16473 1/20 0.43
CHRM2 P08172 1/20 0.42
ADRA2A P08913 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
DRD1 P21728 1/20 0.42
SLC6A2 P23975 1/20 0.42
HTR2A P28223 1/20 0.42
SLC6A4 P31645 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28386447 0.98 CYP2D6 (0.53) CYP2D6CYP2C19DHFRHCN1HCN4
SCHEMBL1921570 0.88 CYP2D6 (0.62) CYP2D6CYP2C19ALDH1A1CYP1A2TSHR
SCHEMBL9381224 0.82 MAPT (0.56) CYP2D6DHFRHCN1HCN4ALDH1A1
SCHEMBL1160956 0.80 DHFR (0.44) CYP2D6CYP2C19DHFRHCN1HCN4
SCHEMBL28470935 0.79 ALDH1A1 (0.53) CYP2D6CYP2C19ALDH1A1NPSR1CYP1A2
SCHEMBL11697719 0.78 CYP2D6 (0.51) CYP2D6CYP2C19ALDH1A1CYP1A2TSHR
SCHEMBL10619140 0.78 CYP2D6 (0.47) CYP2D6CYP2C19ALDH1A1MAPTCYP1A2
SCHEMBL4647647 0.77 ALDH1A1 (0.45) CYP2D6CYP2C19ALDH1A1MAPTCYP1A2
SCHEMBL229388 0.77 ALDH1A1 (0.45) CYP2D6CYP2C19ALDH1A1MAPTCYP1A2
SCHEMBL9848430 0.77 CYP2D6 (0.46) CYP2D6CYP2C19ALDH1A1MAPTCRHBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105683180-B NMDA antagonist prodrugs 阿斯利康(瑞典)有限公司 2020-01-21 CN claimed
EP-4279476-A1 METHOD FOR ALKYLATING ACIDIC FUNCTIONAL GROUP CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2023-11-22 EP disclosed
WO-2022149618-A1 METHOD FOR ALKYLATING ACIDIC FUNCTIONAL GROUP 中外製薬株式会社 2022-07-14 WO disclosed
CN-111187202-A NMDA antagonist prodrugs 阿斯利康(瑞典)有限公司 2020-05-22 CN disclosed
CN-111187202-A NMDA antagonist prodrugs 阿斯利康(瑞典)有限公司 2020-05-22 CN disclosed
CN-105683180-B NMDA antagonist prodrugs 阿斯利康(瑞典)有限公司 2020-01-21 CN disclosed
CN-105683180-B NMDA antagonist prodrugs 阿斯利康(瑞典)有限公司 2020-01-21 CN disclosed