SCHEMBL24630443

SCHEMBL24630443

O=C(Nc1ccc(N2CCNCC2)c(Cl)c1)[C@@H]1CCN1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
HPGD P15428 2/20 0.53
TSHR P16473 2/20 0.53
NPY2R P49146 3/20 0.47
KDM4E B2RXH2 1/20 0.47
RECQL P46063 1/20 0.47
MALT1 Q9UDY8 1/20 0.45
CYP2D6 P10635 2/20 0.44
CCR2 P41597 2/20 0.44
KCNH2 Q12809 2/20 0.44
MEN1 O00255 4/20 0.44
LMNA P02545 4/20 0.44
KMT2A Q03164 4/20 0.44
MAPT P10636 4/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
MAPK1 P28482 2/20 0.44
HTT P42858 1/20 0.44
NPC1 O15118 3/20 0.43
TP53 P04637 2/20 0.43
ALOX15 P16050 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24630108 0.88 NPC1 (0.55) ALDH1A1HPGDTSHRNPY2RKDM4E
SCHEMBL15818617 0.80 KDM4E (0.56) ALDH1A1HPGDTSHRKDM4ERECQL
SCHEMBL8150390 0.78 HPGD (0.54) ALDH1A1HPGDTSHRNPY2RMALT1
SCHEMBL24629992 0.75 KDM4E (0.63) ALDH1A1HPGDNPY2RKDM4ERECQL
SCHEMBL31122602 0.74 ALDH1A1 (0.60) ALDH1A1TSHRMALT1KMT2AMAPT
SCHEMBL24630252 0.74 ALDH1A1 (0.73) ALDH1A1HPGDTSHRCYP2D6MEN1
SCHEMBL29769115 0.74 ALDH1A1 (0.73) ALDH1A1HPGDTSHRCYP2D6MEN1
Trifluoroacetic Acid SCHEMBL7522281 0.74 ALDH1A1 (0.49) ALDH1A1HPGDTSHRNPY2RMALT1
SCHEMBL2531810 0.73 GRM4 (0.66) ALDH1A1MAPTSMN1; SMN2CYP2C19
SCHEMBL27628316 0.73 TSHR (0.53) ALDH1A1HPGDTSHRMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022150574-A1 INHIBITORS OF MYCOBACTERIUM TUBERCULOSIS LIPOAMIDE DEHYDROGENASE CORNELL UNIVERSITY (US) 2022-07-14 WO disclosed