SCHEMBL24632523

SCHEMBL24632523

CNC(=O)NC1CCC(c2ccc(C)cc2F)CC1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
GCK P35557 1/20 0.41
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 1/20 0.40
EPHX1 P07099 1/20 0.40
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
TAS1R2 Q8TE23 1/20 0.39
DRD4 P21917 1/20 0.38
OPRL1 P41146 2/20 0.38
PDE4B Q07343 1/20 0.38
TRPV1 Q8NER1 4/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24632522 0.86 HTR2A (0.42) NPC1RAB9AMEN1KMT2ATAS1R3
SCHEMBL25085619 0.83 SMN1; SMN2 (0.45) NPC1RAB9AGCKMEN1ALDH1A1
SCHEMBL21267605 0.83 PDE2A (0.43) GCKMEN1ALDH1A1KMT2AEPHX1
SCHEMBL24632926 0.81 OPRL1 (0.40) DRD4OPRL1
SCHEMBL16962148 0.79 SLC6A2 (0.43) DRD4OPRL1
SCHEMBL24632526 0.75 HCRTR2 (0.43) ALDH1A1KMT2A
SCHEMBL18503369 0.73 SLC6A2 (0.39) TAS1R3TAS1R1TAS1R2DRD4OPRL1
SCHEMBL13499926 0.72 PTGDR2 (0.42) NPC1RAB9ADRD4OPRL1
SCHEMBL14864497 0.71 PTGDR2 (0.44) NPC1RAB9AOPRL1LMNA
SCHEMBL10282411 0.71 TAS1R3 (0.62) NPC1RAB9AMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022236253-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS NUVATION BIO INC. (US) 2022-11-10 WO disclosed
WO-2022236256-A1 HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS NUVATION BIO INC. (US) 2022-11-10 WO disclosed