SCHEMBL24633971

SCHEMBL24633971

Cc1cc(Br)cc(F)c1C(F)F

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24633970 0.86 CA1 (0.36) CA1CA2
SCHEMBL18099486 0.84 DGAT1 (0.31)
SCHEMBL17420920 0.79 GABRA1 (0.33) CA1CA2
SCHEMBL24633968 0.78 POLB (0.35) CA1CA2
SCHEMBL22805144 0.76 NMT1 (0.34)
SCHEMBL1630637 0.74 ERN1 (0.36)
SCHEMBL26084697 0.74 CA1 (0.31) CA1CA2
SCHEMBL5305665 0.72 HDAC1 (0.35)
SCHEMBL12986534 0.72 GABRA1 (0.41)
SCHEMBL13550059 0.72 NQO2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4309741-A1 CYCLIC COMPOUND HAVING INHIBITORY EFFECT SELECTIVE FOR KRAS BUT NOT FOR HRAS AND NRAS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2024-01-24 EP disclosed
WO-2023214576-A1 CYCLIC COMPOUND HAVING SELECTIVE KRAS INHIBITORY EFFECT ON HRAS AND NRAS 中外製薬株式会社 2023-11-09 WO disclosed
WO-2022234853-A1 CYCLIC COMPOUND HAVING INHIBITORY EFFECT SELECTIVE FOR KRAS BUT NOT FOR HRAS AND NRAS 中外製薬株式会社 2022-11-10 WO disclosed