SCHEMBL2463527

SCHEMBL2463527

CC(C)(C)C(C(N)=O)n1c(C2CCCC2)nc2ccc(N3CCCNCC3)cc2c1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
IDO2 Q6ZQW0 1/20 0.38
PDE7A Q13946 5/20 0.37
PDE7B Q9NP56 2/20 0.37
PDE4D Q08499 1/20 0.37
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
HTR2C P28335 1/20 0.36
MCHR1 Q99705 1/20 0.36
CDK4 P11802 4/20 0.35
CCND1 P24385 4/20 0.35
CCND2 P30279 3/20 0.35
CCND3 P30281 3/20 0.35
NCF1 P14598 1/20 0.34
KCNH2 Q12809 1/20 0.34
HRH4 Q9H3N8 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
KHK P50053 1/20 0.34
ITGB3 P05106 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2466503 0.78 AVPR1B (0.42) IDO1TDO2IDO2PDE7APDE7B
SCHEMBL12334743 0.77 AVPR1B (0.42) KDM4EALDH1A1MAPTHPGD
SCHEMBL4060343 0.70 HTR1A (0.43) HTR1AHTR7HTR2B
SCHEMBL3056004 0.65 ENPP2 (0.47)
SCHEMBL5804762 0.65 MAPK14 (0.44)
SCHEMBL2462426 0.65 AVPR1B (0.60)
SCHEMBL2462438 0.63 AVPR1B (0.44)
SCHEMBL296197 0.60 ENPP2 (0.49)
SCHEMBL30202377 0.60 ENPP2 (0.49)
SCHEMBL1919522 0.60 ENPP2 (0.44) IDO1TDO2IDO2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2069315-B1 QUINAZOLINONE AND ISOQUINOLINONE ACETAMIDE DERIVATIVES ORGANON NV (NL) 2011-09-07 EP disclosed