SCHEMBL24639259

SCHEMBL24639259

CCN1CCN2c3nc(N)c(Cl)cc3OCC[C@H]2C1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 2/20 0.39
KCNH2 Q12809 3/20 0.32
OPRL1 P41146 1/20 0.32
TIPARP Q7Z3E1 8/20 0.32
CHRNA7 P36544 1/20 0.31
HTR3A P46098 1/20 0.31
HTT P42858 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
CYP2D6 P10635 2/20 0.30
CYP2C9 P11712 2/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C19 P33261 1/20 0.30
CYP2C8 P10632 1/20 0.30
SOS1 Q07889 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24639248 1.00 NLRP3 (0.39) NLRP3KCNH2OPRL1TIPARPCHRNA7
SCHEMBL24640720 0.89 OPRL1 (0.33) NLRP3KCNH2OPRL1
SCHEMBL24640631 0.85 SOS1 (0.35) KCNH2CHRNA7HTR3AHRH4SOS1
SCHEMBL24639268 0.85 NLRP3 (0.40) NLRP3TIPARPSOS1
SCHEMBL24640606 0.82 SOS1 (0.39) KCNH2TIPARPCHRNA7HTR3ASOS1
SCHEMBL24640827 0.76 NLRP3 (0.42) NLRP3KCNH2TIPARPCYP2D6CYP2C9
SCHEMBL31245005 0.76 HTR2C (0.44)
SCHEMBL31245376 0.76 HTR2C (0.44)
SCHEMBL31244786 0.76 HTR2C (0.44)
SCHEMBL24639251 0.73 NLRP3 (0.41) NLRP3KCNH2TIPARPCYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022170974-A1 TRICYCLIC DERIVATIVES USEFUL AS PARP7 INHIBITORS JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2022-08-18 WO disclosed