SCHEMBL2464016

SCHEMBL2464016

Clc1ccc(-c2cn(C3CCCCO3)c3ccncc23)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 3/20 0.43
CDK2 P24941 2/20 0.43
DYRK1A Q13627 3/20 0.42
GSK3B P49841 2/20 0.42
NLRP3 Q96P20 1/20 0.39
CYP1A2 P05177 1/20 0.37
TSHR P16473 1/20 0.37
ACVRL1 P37023 1/20 0.35
ACVR1 Q04771 1/20 0.35
KCNH2 Q12809 1/20 0.34
NFATC1 O95644 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
GFER P55789 1/20 0.32
YTHDC1 Q96MU7 1/20 0.32
AKT1 P31749 1/20 0.32
RXRA P19793 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12327177 0.80 DYRK1A (0.66) CDC7CDK2DYRK1AGSK3BNLRP3
SCHEMBL2464056 0.78 DYRK1A (0.57) CDC7CDK2DYRK1AGSK3BACVR1
SCHEMBL12327008 0.75 DYRK1A (0.47) CDC7CDK2DYRK1AGSK3BKCNH2
SCHEMBL18976877 0.74 DYRK1A (0.46) CDC7CDK2DYRK1AGSK3BKCNH2
SCHEMBL1648134 0.71 CYP4F2 (0.41) ALDH1A1GAAMAPTAKT1RXRA
SCHEMBL2464307 0.71 DYRK1A (0.43) CDC7CDK2DYRK1AGSK3BKCNH2
SCHEMBL2468525 0.69 DYRK1A (0.50) CDC7CDK2DYRK1AGSK3BNLRP3
SCHEMBL27926310 0.67 DYRK1A (0.39) CDC7CDK2DYRK1AGSK3BKCNH2
SCHEMBL12327702 0.66 PRKCG (0.49) HPGD
SCHEMBL29281211 0.66 METAP2 (0.34) ACVRL1ACVR1ALDH1A1HPGDYTHDC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2547677-A2 INHIBITORS OF SEMICARABAZIDE - SENSITIVE AMINE OXIDASE Proximagen Limited (GB) 2013-01-23 EP disclosed
WO-2011113798-A2 NEW ENZYME INHIBITOR COMPOUNDS PROXIMAGEN LIMITED (GB) 2011-09-22 WO disclosed