SCHEMBL24640313

SCHEMBL24640313

CC(C)N1CCN2c3ncc(C(F)(F)F)nc3OCCC2C1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 1/20 0.36
TIPARP Q7Z3E1 10/20 0.33
PARP2 Q9UGN5 3/20 0.33
HRH3 Q9Y5N1 3/20 0.32
CHRM2 P08172 1/20 0.31
HTR1A P08908 1/20 0.31
DRD3 P35462 1/20 0.31
HTR2B P41595 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26958161 0.85 HTR2A (0.40) SOS1TIPARPPARP2HTR2B
SCHEMBL24640930 0.84 SOS1 (0.35) SOS1TIPARP
SCHEMBL26958276 0.81 HRH3 (0.33) SOS1HRH3HTR2B
SCHEMBL24639389 0.79 TIPARP (0.49) SOS1TIPARPPARP2CHRM2HTR1A
SCHEMBL24639352 0.79 TIPARP (0.49) SOS1TIPARPPARP2CHRM2HTR1A
SCHEMBL24639355 0.79 TIPARP (0.49) SOS1TIPARPPARP2CHRM2HTR1A
SCHEMBL24639880 0.77 HRH3 (0.31) HRH3
SCHEMBL31245317 0.76 HTR2A (0.44) HTR2B
SCHEMBL29842014 0.76 HTR2A (0.44) HTR2B
SCHEMBL29842130 0.76 HSD11B1 (0.38) CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022170974-A1 TRICYCLIC DERIVATIVES USEFUL AS PARP7 INHIBITORS JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2022-08-18 WO disclosed