Deracoxib

Deracoxib

SCHEMBL24645

COc1ccc(-c2cc(C(F)F)nn2-c2ccc(S(N)(=O)=O)cc2)cc1F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 19/20 1.00
PTGS1 P23219 12/20 1.00
ABCB11 O95342 1/20 1.00
ALDH1A1 P00352 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Deracoxib SCHEMBL29593653 1.00 PTGS2 (1.00) PTGS2PTGS1ABCB11ALDH1A1
Deracoxib SCHEMBL6601340 0.99 PTGS2 (0.98) PTGS2PTGS1ABCB11ALDH1A1
Deracoxib SCHEMBL28723602 0.99 PTGS2 (0.98) PTGS2PTGS1ABCB11ALDH1A1
Deracoxib SCHEMBL6599167 0.95 PTGS2 (0.91) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6343102 0.92 PTGS2 (0.84) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6341965 0.91 PTGS2 (0.83) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6349615 0.90 PTGS2 (0.81) PTGS2PTGS1ABCB11ALDH1A1
Deracoxib SCHEMBL6909431 0.89 PTGS2 (0.80) PTGS2PTGS1ABCB11ALDH1A1
Deracoxib SCHEMBL6598846 0.89 PTGS2 (0.79) PTGS2PTGS1ABCB11ALDH1A1
Deracoxib SCHEMBL6598844 0.89 PTGS2 (0.79) PTGS2PTGS1ABCB11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 7106 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4744663-A2 SKIN COMPOSITION Eaderm Co., Ltd. (JP) 2026-05-20 EP claimed
US-20260000741-A1 METHOD OF AMELIORATING A PRO-INFLAMMATORY IMMUNOPHENOTYPE IN FARBER DISEASE SUBJECTS BY REPEATED ADMINISTRATION OF A RECOMBINANT HUMAN ACID CERAMIDASE ACERAGEN INC (US) 2026-01-01 US claimed
US-12478609-B2 Combination therapies using immuno-DASH inhibitors and PGE2 antagonists TRUSTEES OF TUFTS COLLEGE (US) 2025-11-25 US claimed
EP-4615506-A1 USE OF GSK-3 ACTIVATIOR TO MODULATE PROTEASOME ACTIVITY TO PREVENT AGEING ASSOCIATED CONDITIONS AND DISEASES Sahin, Fikret (TR) 2025-09-17 EP claimed
WO-2025031979-A1 USE OF RIMCAZOLE TO TREAT CANCER KYREXA LTD (GB) 2025-02-13 WO claimed
WO-2024258363-A1 USE OF GSK-3 ACTIVATIOR TO MODULATE PROTEASOME ACTIVITY TO PREVENT AGEING ASSOCIATED CONDITIONS AND DISEASES SAHIN FIKRET (TR) 2024-12-19 WO claimed
US-20240277659-A1 COMBINATION THERAPIES USING IMMUNO-DASH INHIBITORS AND PGE2 ANTAGONISTS TRUSTEES OF TUFTS COLLEGE 2024-08-22 US claimed
CN-118409014-A Detection method of nonsteroidal anti-inflammatory drugs in horse urine 武汉商学院 2024-07-30 CN claimed
CN-118079006-A Skin composition 国立大学法人东京医科齿科大学 2024-05-28 CN claimed
US-11957657-B2 Combination therapies using immuno-dash inhibitors and PGE2 antagonists TRUSTEES OF TUFTS COLLEGE (US) 2024-04-16 US claimed
WO-1997029776-A1 COMBINATIONS HAVING IMMUNOSUPPRESSIVE EFFECTS, CONTAINING CYCLOOXYGENASE-2-INHIBITORS AND 5-LIPOXYGENASE INHIBITORS G.D. SEARLE & CO. (US) 1997-08-21 WO claimed
WO-1997011704-A1 SUBSTITUTED PYRAZOLYL BENZENESULFONAMIDES FOR USE IN VETERINARY THERAPIES AS ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1997-04-03 WO claimed
CN-1141630-A Substituted pyrazolyl benzenesulfonamides for treating inflammation SEARLE & CO (US) 1997-01-29 CN claimed
WO-1996041645-A1 COMBINATION OF A CYCLOOXYGENASE-2 INHIBITOR AND A LEUKOTRIENE B4 RECEPTOR ANTAGONIST FOR THE TREATMENT OF INFLAMMATIONS G.D. SEARLE & CO. (US) 1996-12-27 WO claimed
WO-1996041626-A1 COMPOSITIONS COMPRISING A CYCLOOXYGENASE-2 INHIBITOR AND A 5-LIPOXYGENASE INHIBITOR G.D. SEARLE & CO. (US) 1996-12-27 WO claimed
WO-1996041625-A1 COMPOSITIONS COMPRISING A CYCLOOXYGENASE-2 INHIBITOR AND A LEUKOTRIENE A4 HYDROLASE INHIBITOR G.D. SEARLE & CO. (US) 1996-12-27 WO claimed
WO-1996037476-A1 METHOD OF PREPARING 3-HALOALKYL-1H-PYRAZOLES G.D. SEARLE & CO. (US) 1996-11-28 WO claimed
EP-0731795-A1 SUBSTITUTED PYRAZOLYL BENZENESULFONAMIDES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-09-18 EP claimed
US-5521207-A Substituted pyrazolyl benzenesulfonamide for the treatment of inflammation G.D. SEARLE & CO. (US) 1996-05-28 US claimed
WO-1995015316-A1 SUBSTITUTED PYRAZOLYL BENZENESULFONAMIDES FOR THE TREATMENT OF INFLAMMATION G. D. SEARLE & CO. (US) 1995-06-08 WO claimed