SCHEMBL2464709

SCHEMBL2464709

O=[N+]([O-])c1ccc(Br)nc1Nc1ccccc1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
MYC P01106 1/20 0.42
MAX P61244 1/20 0.42
EPHX2 P34913 1/20 0.41
PTK2 Q05397 1/20 0.41
FGFR4 P22455 1/20 0.40
AURKA O14965 2/20 0.39
AKR1B1 P15121 1/20 0.39
AKR1C4 P17516 1/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
AKR1C1 Q04828 1/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
MAPT P10636 2/20 0.39
GAA P10253 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
TDP1 Q9NUW8 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2194289 0.85 ALDH1A1 (0.46) ALDH1A1MYCMAXEPHX2PTK2
SCHEMBL12335645 0.77 ALDH1A1 (0.40) ALDH1A1MYCMAXEPHX2PTK2
SCHEMBL2572184 0.76 GSK3B (0.58) ALDH1A1MYCAURKAMEN1KMT2A
SCHEMBL18077187 0.76 ALDH1A1 (0.33) ALDH1A1MYCMAXMEN1KMT2A
SCHEMBL2464808 0.75 KIF11 (0.54) FGFR4AURKAAKR1B1AKR1C4AKR1C3
SCHEMBL18077243 0.75 PRKCQ (0.33) ALDH1A1MYCMAXPTK2MEN1
SCHEMBL20529668 0.74 MAPT (0.42) ALDH1A1FGFR4MEN1KMT2AMAPT
SCHEMBL20089577 0.74 ALDH1A1 (0.32) ALDH1A1MYCMAXPRKCQ
SCHEMBL18077191 0.73 ALDH1A1 (0.33) ALDH1A1MYCMAXMAPTSMN1; SMN2
SCHEMBL18077190 0.72 ALDH1A1 (0.32) ALDH1A1MYCMAXMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011116176-A1 3-SUBSTITUED IMIDAZO (4, 5-B) PYRIDINES AND ANALOGS AS SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS INC. (US) 2011-09-22 WO disclosed
WO-2011116176-A1 3-SUBSTITUED IMIDAZO (4, 5-B) PYRIDINES AND ANALOGS AS SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS INC. (US) 2011-09-22 WO disclosed