SCHEMBL2465616

SCHEMBL2465616

Fc1ccc(COc2cccc(Nc3nccn4c(C5CCC5)ncc34)c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 12/20 0.54
F10 P00742 4/20 0.43
MCHR1 Q99705 2/20 0.43
F2 P00734 1/20 0.42
ELANE P08246 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2515230 0.83 IGF1R (0.51) IGF1R
SCHEMBL6014692 0.82 IGF1R (0.45) IGF1RF10
SCHEMBL5400222 0.79 IGF1R (0.43) IGF1R
SCHEMBL5078897 0.72 TNK2 (0.40) IGF1R
SCHEMBL13504863 0.72 TNK2 (0.53)
SCHEMBL2460643 0.71 IGF1R (0.75) IGF1R
SCHEMBL2457076 0.70 IGF1R (1.00) IGF1R
SCHEMBL5083550 0.66 IGF1R (0.40) IGF1R
SCHEMBL5082928 0.66 IGF1R (0.40) IGF1R
SCHEMBL5086159 0.66 TNK2 (0.35) IGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1675860-B1 IMIDAZO[1,5-A]PYRAZINES AS TYROSINE KINASE INHIBITORS OSI PHARM INC (US) 2011-09-21 EP disclosed