SCHEMBL24670154

SCHEMBL24670154

Cc1cc(NC(=O)c2ccc3c(c2)CN(C(=O)OC(C)(C)C)CC3)ccc1C1=CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.52
NR1H2 P55055 1/20 0.49
SCN9A Q15858 2/20 0.46
ESR2 Q92731 1/20 0.45
TMPRSS2 O15393 2/20 0.44
PDK4 Q16654 1/20 0.44
JAK1 P23458 1/20 0.43
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
RAF1 P04049 1/20 0.41
BRAF P15056 1/20 0.41
GRM5 P41594 1/20 0.41
GRM1 Q13255 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
WNT3A P56704 1/20 0.40
IGF1R P08069 1/20 0.40
GRAMD1A Q96CP6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803462 1.00 NAMPT (0.52) NAMPTNR1H2SCN9AESR2TMPRSS2
SCHEMBL29803443 0.96 NAMPT (0.54) NAMPTNR1H2SCN9AESR2TMPRSS2
SCHEMBL29803577 0.96 NAMPT (0.55) NAMPTNR1H2SCN9AESR2TMPRSS2
SCHEMBL24671234 0.96 NAMPT (0.55) NAMPTNR1H2SCN9AESR2TMPRSS2
SCHEMBL29803764 0.92 NAMPT (0.53) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL24670716 0.92 NAMPT (0.53) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL24670163 0.89 NAMPT (0.51) NAMPTNR1H2SCN9AESR2TMPRSS2
SCHEMBL29803391 0.89 NAMPT (0.51) NAMPTNR1H2SCN9AESR2TMPRSS2
SCHEMBL24670852 0.88 NAMPT (0.49) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL24670838 0.88 NAMPT (0.49) NAMPTSCN9APDK4JAK1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed