SCHEMBL24670163

SCHEMBL24670163

CC(C)(C)OC(=O)N1CC=C(c2ccc(C(=O)Nc3ccc4c(c3)CN(C(=O)OC(C)(C)C)CC4)cc2F)CC1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.51
NR1H2 P55055 1/20 0.48
SCN9A Q15858 1/20 0.45
NPC1 O15118 2/20 0.45
ESR2 Q92731 1/20 0.45
TMPRSS2 O15393 2/20 0.44
RAB9A P51151 1/20 0.44
PDK4 Q16654 1/20 0.44
JAK1 P23458 1/20 0.42
GRM5 P41594 3/20 0.42
GRM1 Q13255 3/20 0.42
CDK9 P50750 1/20 0.41
WDR5 P61964 1/20 0.41
MAPK14 Q16539 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29803391 1.00 NAMPT (0.51) NAMPTNR1H2SCN9ANPC1ESR2
SCHEMBL24671531 0.96 NAMPT (0.54) NAMPTNR1H2SCN9ANPC1ESR2
SCHEMBL29803468 0.96 NAMPT (0.54) NAMPTNR1H2SCN9ANPC1ESR2
SCHEMBL29803696 0.92 NAMPT (0.52) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL24669339 0.92 NAMPT (0.52) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL24670154 0.89 NAMPT (0.52) NAMPTNR1H2SCN9ANPC1ESR2
SCHEMBL29803462 0.89 NAMPT (0.52) NAMPTNR1H2SCN9ANPC1ESR2
SCHEMBL29803278 0.89 NAMPT (0.49) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL24670852 0.89 NAMPT (0.49) NAMPTSCN9APDK4JAK1GRM5
SCHEMBL24671269 0.88 NAMPT (0.63) NAMPTNR1H2SCN9ANPC1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed