SCHEMBL24670181

SCHEMBL24670181

COc1cc(N2CCC(CO)CC2)ccc1C1CCC(=O)NC1=O

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 15/20 0.43
DDB1 Q16531 13/20 0.43
PDE7A Q13946 1/20 0.42
SUV39H2 Q9H5I1 2/20 0.38
NR3C1 P04150 1/20 0.37
PGR P06401 1/20 0.37
SLC6A4 P31645 1/20 0.37
KCNH2 Q12809 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30066248 1.00 CRBN (0.43) CRBNDDB1PDE7ASUV39H2NR3C1
SCHEMBL31134484 0.87 CRBN (0.55) CRBNDDB1PDE7A
Hydrochloric Acid SCHEMBL27039409 0.86 CRBN (0.54) CRBNDDB1PDE7A
SCHEMBL24670661 0.86 CRBN (0.50) CRBNDDB1
SCHEMBL30066508 0.86 CRBN (0.50) CRBNDDB1
SCHEMBL30801303 0.86 CRBN (0.47) CRBNDDB1
SCHEMBL31722466 0.85 CRBN (0.43) CRBNDDB1NR3C1PGRSLC6A4
SCHEMBL24670182 0.84 CRBN (0.44) CRBNDDB1NR3C1PGRSLC6A4
SCHEMBL30066195 0.84 CRBN (0.44) CRBNDDB1NR3C1PGRSLC6A4
SCHEMBL24670681 0.84 CRBN (0.42) CRBNDDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116261458-B PLK1 degradation inducing compounds 厄普特拉株式会社 2024-05-24 CN disclosed
CN-117693502-A Compounds for inhibiting or degrading ITK, compositions comprising the same, methods of making the same, and methods of using the same 纽力克斯治疗公司 2024-03-12 CN disclosed
US-20230242541-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND UPPTHERA, INC. (KR) 2023-08-03 US disclosed
US-20230242541-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND UPPTHERA, INC. (KR) 2023-08-03 US disclosed
CN-116261458-A Novel PLK1 degradation inducing compounds 厄普特拉株式会社 2023-06-13 CN disclosed
WO-2022235715-A1 COMPOUNDS FOR INHIBITING OR DEGRADING ITK, COMPOSITIONS, COMPRISING THE SAME METHODS OF THEIR MAKING AND METHODS OF THEIR USE NURIX THERAPEUTICS, INC. (US) 2022-11-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230242541-A1 NOVEL PLK1 DEGRADATION INDUCING COMPOUND PLK1, BUB1B, BUB1 CRBN 2136/4885DDB1 132/4885PDE7A 3233/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.