SCHEMBL24670201

SCHEMBL24670201

CCCc1ccc(C(=O)NC)nc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 3/20 0.57
ALDH1A1 P00352 4/20 0.55
KDM4E B2RXH2 3/20 0.55
NFKB1 P19838 2/20 0.55
MEN1 O00255 1/20 0.55
LMNA P02545 1/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
MAPT P10636 1/20 0.55
PKM P14618 1/20 0.55
ALOX15 P16050 1/20 0.55
TSHR P16473 1/20 0.55
THPO P40225 1/20 0.55
BLM P54132 1/20 0.55
PMP22 Q01453 1/20 0.55
KMT2A Q03164 1/20 0.55
HIF1A Q16665 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
PARP1 P09874 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7794120 0.90 NFKB1 (0.69) PLK1ALDH1A1KDM4ENFKB1MEN1
SCHEMBL12561176 0.86 PLK1 (0.55) PLK1ALDH1A1KDM4ENFKB1MEN1
SCHEMBL659153 0.84 P4HTM (0.69) ALDH1A1KDM4ENFKB1MEN1LMNA
SCHEMBL26970993 0.83 PARP1 (0.51) PLK1ALDH1A1KDM4ENFKB1MEN1
SCHEMBL30027907 0.83 PARP1 (0.51) PLK1ALDH1A1KDM4ENFKB1MEN1
SCHEMBL16597438 0.83 PARP1 (0.51) PLK1ALDH1A1KDM4ENFKB1MEN1
SCHEMBL2642502 0.81 PARP1 (0.50) PLK1ALDH1A1KDM4ENFKB1MEN1
SCHEMBL2642500 0.81 PARP1 (0.50) PLK1ALDH1A1KDM4ENFKB1MEN1
SCHEMBL26970992 0.81 PARP1 (0.50) PLK1ALDH1A1KDM4ENFKB1MEN1
SCHEMBL8150967 0.81 ALDH1A1 (0.60) PLK1ALDH1A1KDM4ENFKB1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022235715-A1 COMPOUNDS FOR INHIBITING OR DEGRADING ITK, COMPOSITIONS, COMPRISING THE SAME METHODS OF THEIR MAKING AND METHODS OF THEIR USE NURIX THERAPEUTICS, INC. (US) 2022-11-10 WO disclosed