SCHEMBL24670871

SCHEMBL24670871

CNC(=N)N1CC=C(c2ccc(C(=O)Nc3cc(C)c(C4=CCN(C(=N)N)CC4)c(F)c3)cc2F)CC1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TMPRSS2 O15393 6/20 0.42
CCNT1 O60563 7/20 0.38
CDK9 P50750 7/20 0.38
MAPT P10636 4/20 0.33
TRPV1 Q8NER1 1/20 0.33
BTK Q06187 1/20 0.33
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29802833 0.95 TMPRSS2 (0.46) TMPRSS2CCNT1CDK9MAPTTRPV1
SCHEMBL24670857 0.89 TMPRSS2 (0.45) TMPRSS2CCNT1CDK9MAPTTRPV1
SCHEMBL29803204 0.85 TMPRSS2 (0.52) TMPRSS2MAPTTRPV1POLB
SCHEMBL24671270 0.85 TMPRSS2 (0.52) TMPRSS2MAPTTRPV1POLB
SCHEMBL29803214 0.84 TMPRSS2 (0.52) TMPRSS2MAPTTRPV1
SCHEMBL24670599 0.84 TRPV1 (0.45) TMPRSS2MAPTTRPV1
SCHEMBL24669468 0.83 TMPRSS2 (0.52) TMPRSS2MAPTTRPV1POLB
SCHEMBL24669503 0.81 PDK4 (0.46) CCNT1CDK9
SCHEMBL24669447 0.81 TMPRSS2 (0.48) TMPRSS2MAPT
SCHEMBL29803358 0.80 TMPRSS2 (0.47) TMPRSS2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed