SCHEMBL24670528

SCHEMBL24670528

N=C(N)N1CC=C(c2ccc(NC(=O)c3cc(C4=CCN(C(=N)N)CC4)co3)nc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 12/20 0.46
MAPT P10636 2/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
EGLN1 Q9GZT9 2/20 0.36
TRPV1 Q8NER1 2/20 0.36
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
WNT1 P04628 1/20 0.35
CLK2 P49760 1/20 0.35
CLK3 P49761 1/20 0.35
GSK3B P49841 1/20 0.35
DYRK1A Q13627 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29803709 0.94 NAMPT (0.43) NAMPTMAPTLMNAHTTNPSR1
SCHEMBL24670492 0.86 ALDH1A1 (0.44) NAMPTMAPTLMNAHTTNPC1
SCHEMBL24671065 0.83 NAMPT (0.49) NAMPT
Trifluoroacetic Acid SCHEMBL29803611 0.80 MAPT (0.42) NAMPTMAPTLMNAHTTNPSR1
SCHEMBL24671431 0.79 NAMPT (0.48) NAMPTMAPTLMNAHTTNPSR1
SCHEMBL24671577 0.79 ABCB1 (0.47) NAMPTNPC1RAB9A
SCHEMBL24670508 0.78 MAPT (0.44) MAPTLMNAHTTNPSR1NPC1
SCHEMBL24669855 0.78 MAPT (0.37) NAMPTMAPTLMNAHTTNPSR1
SCHEMBL24891672 0.78 NAMPT (0.43) NAMPTEGLN1ALDH1A1
SCHEMBL30181035 0.78 NAMPT (0.43) NAMPTEGLN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO claimed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed