SCHEMBL24671263

SCHEMBL24671263

O=C(Nc1ccc(C2=CCNCC2)c(Cl)c1)c1ccc(C2=CCNCC2)s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
RXFP1 Q9HBX9 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MAPKAPK2 P49137 2/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
MEN1 O00255 2/20 0.40
NFKB1 P19838 2/20 0.40
NFKB2 Q00653 2/20 0.40
KMT2A Q03164 2/20 0.40
RELA Q04206 2/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
ESRRG P62508 6/20 0.39
ESR1 P03372 4/20 0.39
ESR2 Q92731 2/20 0.39
PRSS12 P56730 1/20 0.37
PPARG P37231 1/20 0.37
NR2E3 Q9Y5X4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL29803663 0.93 KDM4E (0.40) KDM4ERXFP1NPSR1MAPKAPK2NPC1
SCHEMBL24671298 0.87 ESRRG (0.43) KDM4ERXFP1NPSR1MAPKAPK2ESRRG
SCHEMBL24670406 0.85 IMPDH2 (0.45) KDM4EMAPKAPK2SMN1; SMN2KMT2AALDH1A1
SCHEMBL29803733 0.83 MAPKAPK2 (0.52) KDM4ERXFP1MAPKAPK2NPC1RAB9A
Trifluoroacetic Acid SCHEMBL29803840 0.82 MAPT (0.39) KDM4ERXFP1NPSR1NPC1RAB9A
SCHEMBL29803327 0.82 NPC1 (0.52) KDM4EMAPKAPK2NPC1RAB9AMEN1
Hydrochloric Acid SCHEMBL29803461 0.80 TP53 (0.46) KDM4ERXFP1MAPKAPK2NPC1RAB9A
Trifluoroacetic Acid SCHEMBL29803398 0.79 IMPDH2 (0.41) KDM4ESMN1; SMN2KMT2ANCOR2KCNH2
SCHEMBL24670348 0.78 TP53 (0.46) KDM4ERXFP1MAPKAPK2NPC1RAB9A
SCHEMBL29803234 0.78 MAPT (0.44) KDM4ERXFP1NPSR1MAPKAPK2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed
WO-2022192162-A1 NOVEL HETEROAROMATIC COMPOUNDS EXHIBITING ANTIFUNGAL ACTIVITY AND THEIR METHOD OF USE FOX CHASE CHEMICAL DIVERSITY CENTER, INC. (US) 2022-09-15 WO disclosed